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TargetRetinol-binding protein 4
LigandBDBM50347599
Substrate/Competitorn/a
Meas. Tech.ChEMBL_756077 (CHEMBL1804187)
EC50 154±n/a nM
Citation Campos-Sandoval, JARedondo, CKinsella, GKPal, AJones, GEyre, GSHirst, SCFindlay, JB Fenretinide derivatives act as disrupters of interactions of serum retinol binding protein (sRBP) with transthyretin and the sRBP receptor. J Med Chem54:4378-87 (2011) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Retinol-binding protein 4
Name:Retinol-binding protein 4
Synonyms:PRBP | Plasma retinol-binding protein | RBP | RBP4 | RET4_HUMAN | Retinol-binding protein 4 | Retinol-binding protein 4 (RBP4) | spa binding assay for rbp4
Type:Protein
Mol. Mass.:23008.75
Organism:Homo sapiens (Human)
Description:P02753
Residue:201
Sequence:
MKWVWALLLLAALGSGRAERDCRVSSFRVKENFDKARFSGTWYAMAKKDPEGLFLQDNIV
AEFSVDETGQMSATAKGRVRLLNNWDVCADMVGTFTDTEDPAKFKMKYWGVASFLQKGND
DHWIVDTDYDTYAVQYSCRLLNLDGTCADSYSFVFSRDPNGLPPEAQKIVRQRQEELCLA
RQYRLIVHNGYCDGRSERNLL
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  Blast E-value cutoff:
BDBM50347599
n/a
NameBDBM50347599
Synonyms:CHEMBL1802454
TypeSmall organic molecule
Emp. Form.C24H35NO2
Mol. Mass.369.5402
SMILESC\C(\C=C\C1=C(C)CCCC1(C)C)=C/C=C/C(/C)=C/C(=O)N1CCOCC1 |c:4|
Structure
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