| Reaction Details |
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 | Report a problem with these data |
| Target | D(1A) dopamine receptor |
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| Ligand | BDBM50347630 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_755707 (CHEMBL1803209) |
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| Ki | 220±n/a nM |
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| Citation |  Kühhorn, J; Hübner, H; Gmeiner, P Bivalent dopamine D2 receptor ligands: synthesis and binding properties. J Med Chem54:4896-903 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(1A) dopamine receptor |
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| Name: | D(1A) dopamine receptor |
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| Synonyms: | DRD1 | DRD1_PIG | Dopamine D1 receptor |
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| Type: | PROTEIN |
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| Mol. Mass.: | 49269.92 |
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| Organism: | Sus scrofa |
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| Description: | ChEMBL_1460140 |
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| Residue: | 446 |
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| Sequence: | MRTLNTSTMDGTGLVVERDFSFRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTN
FFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVD
RYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTSPSDGNVTSLG
KTTHNCDSSLSRTYAISSSLISFYIPVAIMIVTYTRIYRIAQKQIRRISALERAAVHAKN
CQTTAGNGNPAECSQPESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFILNCMVPFCGS
GETKPFCIDSITFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCYRLCPTSTNAIET
VSINNNGAVVFSSHHEPRGSISKDCNLVYLIPHAVGSSEDLKKEEAGGIASPLEKLSPAL
SVILDYDTDVSLEKIQPITQNGQHPT
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| BDBM50347630 |
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| n/a |
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| Name | BDBM50347630 |
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| Synonyms: | CHEMBL1803024 |
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| Type | Small organic molecule |
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| Emp. Form. | C56H76N10O6 |
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| Mol. Mass. | 985.266 |
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| SMILES | COc1ccccc1N1CCN(Cc2ccc(OCCCc3cn(CCCCCCCCn4cc(CCCOc5ccc(CN6CCN(CC6)c6ccccc6OC)cc5OC)nn4)nn3)c(OC)c2)CC1 |
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| Structure | 
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