| Reaction Details |
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 | Report a problem with these data |
| Target | Prostaglandin F2-alpha receptor |
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| Ligand | BDBM50350366 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_761108 (CHEMBL1815362) |
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| Ki | 1400±n/a nM |
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| Citation |  Iwahashi, M; Shimabukuro, A; Onoda, T; Matsunaga, Y; Okada, Y; Matsumoto, R; Nambu, F; Nakai, H; Toda, M Discovery of selective indole-based prostaglandin D2 receptor antagonist. Bioorg Med Chem19:4574-88 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Prostaglandin F2-alpha receptor |
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| Name: | Prostaglandin F2-alpha receptor |
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| Synonyms: | PF2R_MOUSE | ProstaglandinF2Alpha | Ptgfr |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40714.02 |
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| Organism: | MOUSE |
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| Description: | ProstaglandinF2Alpha PTGFR MOUSE::P43117 |
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| Residue: | 366 |
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| Sequence: | MSMNSSKQPVSPAAGLIANTTCQTENRLSVFFSIIFMTVGILSNSLAIAILMKAYQRFRQ
KSKASFLLLASGLVITDFFGHLINGGIAVFVYASDKDWIRFDQSNILCSIFGISMVFSGL
CPLFLGSAMAIERCIGVTNPIFHSTKITSKHVKMILSGVCMFAVFVAVLPILGHRDYQIQ
ASRTWCFYNTEHIEDWEDRFYLLFFSFLGLLALGVSFSCNAVTGVTLLRVKFRSQQHRQG
RSHHLEMIIQLLAIMCVSCVCWSPFLVTMANIAINGNNSPVTCETTLFALRMATWNQILD
PWVYILLRKAVLRNLYKLASRCCGVNIISLHIWELSSIKNSLKVAAISESPAAEKESQQA
SSEAGL
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| BDBM50350366 |
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| n/a |
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| Name | BDBM50350366 |
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| Synonyms: | CHEMBL1813287 |
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| Type | Small organic molecule |
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| Emp. Form. | C30H30N2O4 |
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| Mol. Mass. | 482.5702 |
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| SMILES | CCN1[C@@H](COc2ccc(C(=O)n3c(C)c(CC(O)=O)c4ccccc34)c(C)c2)Cc2ccccc12 |r| |
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| Structure | 
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