| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Prostaglandin D2 receptor |
|---|
| Ligand | BDBM50152515 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_764675 (CHEMBL1821227) |
|---|
| Ki | 16±n/a nM |
|---|
| Citation |  Iwahashi, M; Takahashi, E; Tanaka, M; Matsunaga, Y; Okada, Y; Matsumoto, R; Nambu, F; Nakai, H; Toda, M Design and synthesis of new prostaglandin D2 receptor antagonists. Bioorg Med Chem19:5361-71 (2011) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Prostaglandin D2 receptor |
|---|
| Name: | Prostaglandin D2 receptor |
|---|
| Synonyms: | PD2R_MOUSE | Prostanoid DP receptor | Ptgdr |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 40018.63 |
|---|
| Organism: | Mus musculus |
|---|
| Description: | ChEMBL_788408 |
|---|
| Residue: | 357 |
|---|
| Sequence: | MNESYRCQTSTWVERGSSATMGAVLFGAGLLGNLLALVLLARSGLGSCRPGPLHPPPSVF
YVLVCGLTVTDLLGKCLISPMVLAAYAQNQSLKELLPASGNQLCETFAFLMSFFGLASTL
QLLAMAVECWLSLGHPFFYQRHVTLRRGVLVAPVVAAFCLAFCALPFAGFGKFVQYCPGT
WCFIQMIHKERSFSVIGFSVLYSSLMALLVLATVVCNLGAMYNLYDMHRRQRHYPHRCSR
DRAQSGSDYRHGSLHPLEELDHFVLLALMTVLFTMCSLPLIYRAYYGAFKLENKAEGDSE
DLQALRFLSVISIVDPWIFIIFRTSVFRMLFHKVFTRPLIYRNWSSHSQQSNVESTL
|
|
|
|---|
| BDBM50152515 |
|---|
| n/a |
|---|
| Name | BDBM50152515 |
|---|
| Synonyms: | CHEMBL364841 | {2-Methyl-1-[4-(4-methyl-3,4-dihydro-2H-benzo[1,4]oxazin-2-ylmethoxy)-benzoyl]-1H-indol-4-yl}-acetic acid |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C28H26N2O5 |
|---|
| Mol. Mass. | 470.5164 |
|---|
| SMILES | CN1C[C@@H](COc2ccc(cc2)C(=O)n2c(C)cc3c(CC(O)=O)cccc23)Oc2ccccc12 |
|---|
| Structure | 
|
|---|
Search and Browse
