| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Transcriptional activator protein TraR |
|---|
| Ligand | BDBM50266163 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_765233 (CHEMBL1827786) |
|---|
| IC50 | 1250±n/a nM |
|---|
| Citation |  Lowery, CA; Salzameda, NT; Sawada, D; Kaufmann, GF; Janda, KD Medicinal chemistry as a conduit for the modulation of quorum sensing. J Med Chem53:7467-89 (2010) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Transcriptional activator protein TraR |
|---|
| Name: | Transcriptional activator protein TraR |
|---|
| Synonyms: | TRAR_RHIRD | traR |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 26741.83 |
|---|
| Organism: | Rhizobium radiobacter |
|---|
| Description: | ChEMBL_765233 |
|---|
| Residue: | 234 |
|---|
| Sequence: | MQHWLDKLTDLAAIEGDECILKTGLADIADHFGFTGYAYLHIQHRHITAVTNYHRQWQST
YFDKKFEALDPVVKRARSRKHIFTWSGEHERPTLSKDERAFYDHASDFGIRSGITIPIKT
ANGFMSMFTMASDKPVIDLDREIDAVAAAATIGQIHARISFLRTTPTAEDAAWLDPKEAT
YLRWIAVGKTMEEIADVEGVKYNSVRVKLREAMKRFDVRSKAHLTALAIRRKLI
|
|
|
|---|
| BDBM50266163 |
|---|
| n/a |
|---|
| Name | BDBM50266163 |
|---|
| Synonyms: | (S)-2-(4-iodophenyl)-N-(2-oxotetrahydrofuran-3-yl)acetamide | CHEMBL468790 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C12H12INO3 |
|---|
| Mol. Mass. | 345.1331 |
|---|
| SMILES | Ic1ccc(CC(=O)N[C@H]2CCOC2=O)cc1 |r| |
|---|
| Structure | 
|
|---|
Search and Browse
