| Reaction Details |
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 | Report a problem with these data |
| Target | Trace amine-associated receptor 1 |
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| Ligand | BDBM50274042 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_792735 (CHEMBL1930650) |
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| EC50 | 2140±n/a nM |
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| Citation |  Lewin, AH; Miller, GM; Gilmour, B Trace amine-associated receptor 1 is a stereoselective binding site for compounds in the amphetamine class. Bioorg Med Chem19:7044-8 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Trace amine-associated receptor 1 |
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| Name: | Trace amine-associated receptor 1 |
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| Synonyms: | TA1 | TAAR1 | TAAR1_MACMU | TAR1 | TRAR1 | TaR-1 | Trace amine receptor 1 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 38812.87 |
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| Organism: | Macaca mulatta |
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| Description: | ChEMBL_792735 |
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| Residue: | 338 |
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| Sequence: | MPFCHNIINISCVKNNWSNDVRASLYSLMALIILTTLVGNLIVIVSISHFKQLHTPTNWL
IHSMATVDFLLGCLVMPYSMVRSAEHCWYFGEVFCKIHTSTDIMLSSASIFHLSFISIDR
YYAVCDPLRYKAKINILVVCVMIFISWSVPAVFAFGMIFLELNFKGAEEIYYKHVHCRGG
CSVFFSKISGVLAFMTSFYIPGSIMLCIYYRIYLIAKEQARSINDANQKLQIGLEMKNGI
SQSKERKAVKTLGIVMGVFLICWCPFFVCTVIDPFLHYTIPPTLNDVLIWFGYLNSTFNP
MVYAFFYPWFRKALKMILFGKIFQKDSSRCKLFLESSS
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| BDBM50274042 |
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| n/a |
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| Name | BDBM50274042 |
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| Synonyms: | (S)-1-(4-bromo-2,5-dimethoxyphenyl)propan-2-amine | CHEMBL468880 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H16BrNO2 |
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| Mol. Mass. | 274.154 |
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| SMILES | COc1cc(C[C@H](C)N)c(OC)cc1Br |r| |
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| Structure | 
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