| Reaction Details |
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 | Report a problem with these data |
| Target | Sigma non-opioid intracellular receptor 1 |
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| Ligand | BDBM50359593 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_792760 (CHEMBL1930675) |
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| Ki | 14690±n/a nM |
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| Citation |  Hajipour, AR; Guo, LW; Pal, A; Mavlyutov, T; Ruoho, AE Electron-donating para-methoxy converts a benzamide-isoquinoline derivative into a highly Sigma-2 receptor selective ligand. Bioorg Med Chem19:7435-40 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Sigma non-opioid intracellular receptor 1 |
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| Name: | Sigma non-opioid intracellular receptor 1 |
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| Synonyms: | Opioid receptor | Oprs1 | SGMR1_RAT | Sigma | Sigma non-opioid intracellular receptor 1 | Sigma opioid receptor | Sigma-1 | Sigmar1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 25266.54 |
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| Organism: | RAT |
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| Description: | Q9R0C9 |
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| Residue: | 223 |
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| Sequence: | MPWAVGRRWAWITLFLTIVAVLIQAVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSHGHSGRY
WAEISDTIISGTFHQWREGTTKSEVYYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALSDTIFSTQDFLTLFYTLRAYARGLRLELTTYLFGQDP
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| BDBM50359593 |
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| n/a |
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| Name | BDBM50359593 |
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| Synonyms: | CHEMBL1927700 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H27N3O5 |
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| Mol. Mass. | 413.4669 |
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| SMILES | COc1cc2CCN(CCCCNC(=O)c3ccc(cc3)[N+]([O-])=O)Cc2cc1OC |
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| Structure | 
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