| Reaction Details |
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 | Report a problem with these data |
| Target | Prostaglandin E2 receptor EP3 subtype |
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| Ligand | BDBM50360151 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_793559 (CHEMBL1932310) |
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| Ki | 1800±n/a nM |
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| Citation |  Kambe, T; Maruyama, T; Nagase, T; Ogawa, S; Minamoto, C; Sakata, K; Maruyama, T; Nakai, H; Toda, M Synthesis and evaluation of novel modified¿-lactam prostanoids as EP4 subtype-selective agonists. Bioorg Med Chem20:702-13 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Prostaglandin E2 receptor EP3 subtype |
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| Name: | Prostaglandin E2 receptor EP3 subtype |
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| Synonyms: | PE2R3_MOUSE | PGE receptor, EP3 isoform alpha | Prostaglandin E2 receptor EP3 isoform alpha | Prostaglandin E3 | Prostanoid EP3 receptor | Ptger3 | Ptgerep3 |
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| Type: | G-protein coupled receptor |
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| Mol. Mass.: | 40092.50 |
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| Organism: | Mus musculus (Mouse) |
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| Description: | n/a |
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| Residue: | 365 |
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| Sequence: | MASMWAPEHSAEAHSNLSSTTDDCGSVSVAFPITMMVTGFVGNALAMLLVSRSYRRRESK
RKKSFLLCIGWLALTDLVGQLLTSPVVILVYLSQRRWEQLDPSGRLCTFFGLTMTVFGLS
SLLVASAMAVERALAIRAPHWYASHMKTRATPVLLGVWLSVLAFALLPVLGVGRYSVQWP
GTWCFISTGPAGNETDPAREPGSVAFASAFACLGLLALVVTFACNLATIKALVSRCRAKA
AVSQSSAQWGRITTETAIQLMGIMCVLSVCWSPLLIMMLKMIFNQMSVEQCKTQMGKEKE
CNSFLIAVRLASLNQILDPWVYLLLRKILLRKFCQIRDHTNYASSSTSLPCPGSSALMWS
DQLER
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| BDBM50360151 |
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| n/a |
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| Name | BDBM50360151 |
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| Synonyms: | CHEMBL1929543 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H24FNO4S2 |
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| Mol. Mass. | 413.527 |
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| SMILES | O[C@@H](Cc1cccc(F)c1)\C=C\[C@H]1CSC(=O)N1CCSCCCC(O)=O |r| |
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| Structure | 
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