| Reaction Details |
|---|
 | Report a problem with these data |
| Target | B2 bradykinin receptor |
|---|
| Ligand | BDBM50286392 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEBML_40427 |
|---|
| Ki | 770±n/a nM |
|---|
| Citation |  Salvino, JM; Seoane, PR; Douty, BD; Awad, MA; Hoyer, D; Ross, TM; Dolle, RE; Houck, WT; Faunce, DM; Sawutz, DG Structure activity relationships of non-peptide bradykinin B2 receptor antagonists Bioorg Med Chem Lett5:357-362 (1995) Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| B2 bradykinin receptor |
|---|
| Name: | B2 bradykinin receptor |
|---|
| Synonyms: | B2 BRADYKININ | B2 bradykinin receptor | B2R | BDKRB2 | BK-2 receptor | BKR2 | BKRB2_HUMAN | Bradykinin B2 receptor |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 44467.17 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | B2 BRADYKININ BDKRB2 HUMAN::P30411 |
|---|
| Residue: | 391 |
|---|
| Sequence: | MFSPWKISMFLSVREDSVPTTASFSADMLNVTLQGPTLNGTFAQSKCPQVEWLGWLNTIQ
PPFLWVLFVLATLENIFVLSVFCLHKSSCTVAEIYLGNLAAADLILACGLPFWAITISNN
FDWLFGETLCRVVNAIISMNLYSSICFLMLVSIDRYLALVKTMSMGRMRGVRWAKLYSLV
IWGCTLLLSSPMLVFRTMKEYSDEGHNVTACVISYPSLIWEVFTNMLLNVVGFLLPLSVI
TFCTMQIMQVLRNNEMQKFKEIQTERRATVLVLVVLLLFIICWLPFQISTFLDTLHRLGI
LSSCQDERIIDVITQIASFMAYSNSCLNPLVYVIVGKRFRKKSWEVYQGVCQKGGCRSEP
IQMENSMGTLRTSISVERQIHKLQDWAGSRQ
|
|
|
|---|
| BDBM50286392 |
|---|
| n/a |
|---|
| Name | BDBM50286392 |
|---|
| Synonyms: | Bis-[4-(tripentyl-lambda*5*-phosphanylmethyl)-phenyl]-methanone; dichloride | CHEMBL121565 | Tripentyl-[6-(tripentyl-lambda*5*-phosphanylmethyl)-naphthalen-2-ylmethyl]-phosphonium; dichloride |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C45H78OP2 |
|---|
| Mol. Mass. | 697.0466 |
|---|
| SMILES | CCCCC[P+](CCCCC)(CCCCC)Cc1ccc(cc1)C(=O)c1ccc(C[P+](CCCCC)(CCCCC)CCCCC)cc1 |
|---|
| Structure | 
|
|---|
Search and Browse
