| Reaction Details |
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 | Report a problem with these data |
| Target | Glycerol kinase |
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| Ligand | BDBM18135 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_72907 |
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| Ki | 300000±n/a nM |
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| Citation |  Bystrom, CE; Pettigrew, DW; Remington, S; Branchaud, BP ATP analogs with non-transferable groups in the position as inhibitors of glycerol kinase Bioorg Med Chem Lett7:2613-2616 (1997) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Glycerol kinase |
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| Name: | Glycerol kinase |
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| Synonyms: | GK | GLPK_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 61243.96 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_72907 |
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| Residue: | 559 |
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| Sequence: | MAASKKAVLGPLVGAVDQGTSSTRFLVFNSKTAELLSHHQVEIKQEFPREGWVEQDPKEI
LHSVYECIEKTCEKLGQLNIDISNIKAIGVSNQRETTVVWDKITGEPLYNAVVWLDLRTQ
STVESLSKRIPGNNNFVKSKTGLPLSTYFSAVKLRWLLDNVRKVQKAVEEKRALFGTIDS
WLIWSLTGGVNGGVHCTDVTNASRTMLFNIHSLEWDKQLCEFFGIPMEILPNVRSSSEIY
GLMKISHSVKAGALEGVPISGCLGDQSAALVGQMCFQIGQAKNTYGTGCFLLCNTGHKCV
FSDHGLLTTVAYKLGRDKPVYYALEGSVAIAGAVIRWLRDNLGIIKTSEEIEKLAKEVGT
SYGCYFVPAFSGLYAPYWEPSARGIICGLTQFTNKCHIAFAALEAVCFQTREILDAMNRD
CGIPLSHLQVDGGMTSNKILMQLQADILYIPVVKPSMPETTALGAAMAAGAAEGVGVWSL
EPEDLSAVTMERFEPQINAEESEIRYSTWKKAVMKSMGWVTTQSPESGDPSIFCSLPLGF
FIVSSMVMLIGARYISGIP
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| BDBM18135 |
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| n/a |
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| Name | BDBM18135 |
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| Synonyms: | ({[({[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy}(hydroxy)phosphoryl)oxy](hydroxy)phosphoryl}methyl)phosphonic acid | AMPPCP | ATP,Beta Gamma-me | CHEMBL133463 | adenylylmethylenediphosphonate |
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| Type | Nucleoside or nucleotide |
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| Emp. Form. | C11H18N5O12P3 |
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| Mol. Mass. | 505.2082 |
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| SMILES | Nc1ncnc2n(cnc12)[C@@H]1O[C@H](COP(O)(=O)OP(O)(=O)CP(O)(O)=O)[C@@H](O)[C@H]1O |r| |
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| Structure | 
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