| Reaction Details |
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 | Report a problem with these data |
| Target | 4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5 |
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| Ligand | BDBM92459 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_69264 |
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| IC50 | 67000±n/a nM |
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| Citation |  Schuster, M; Blechert, S Inhibition of fucosyltransferase V by a GDP-Azasugar. Bioorg Med Chem Lett11:1809-11 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| 4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5 |
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| Name: | 4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5 |
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| Synonyms: | FUT5 | FUT5_HUMAN | Fucosyltransferase 5 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 43016.71 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_69264 |
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| Residue: | 374 |
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| Sequence: | MDPLGPAKPQWLWRRCLAGLLFQLLVAVCFFSYLRVSRDDATGSPRPGLMAVEPVTGAPN
GSRCQDSMATPAHPTLLILLWTWPFNTPVALPRCSEMVPGAADCNITADSSVYPQADAVI
VHHWDIMYNPSANLPPPTRPQGQRWIWFSMESPSNCRHLEALDGYFNLTMSYRSDSDIFT
PYGWLEPWSGQPAHPPLNLSAKTELVAWAVSNWKPDSARVRYYQSLQAHLKVDVYGRSHK
PLPKGTMMETLSRYKFYLAFENSLHPDYITEKLWRNALEAWAVPVVLGPSRSNYERFLPP
DAFIHVDDFQSPKDLARYLQELDKDHARYLSYFRWRETLRPRSFSWALAFCKACWKLQQE
SRYQTVRSIAAWFT
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| BDBM92459 |
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| n/a |
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| Name | BDBM92459 |
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| Synonyms: | CHEMBL384759 | GDP | Guanosine Diphosphate |
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| Type | Small molecule |
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| Emp. Form. | C10H15N5O11P2 |
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| Mol. Mass. | 443.2005 |
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| SMILES | Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H](COP(O)(=O)OP(O)(O)=O)[C@@H](O)[C@H]1O |
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| Structure | 
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