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TargetProtein Tat
LigandBDBM50097336
Substrate/Competitorn/a
Meas. Tech.ChEMBL_209907 (CHEMBL811911)
Kd 290±n/a nM
Citation Hamasaki, KUeno, A Aminoglycoside antibiotics, neamine and its derivatives as potent inhibitors for the RNA-protein interactions derived from HIV-1 activators. Bioorg Med Chem Lett11:591-4 (2001) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Protein Tat
Name:Protein Tat
Synonyms:Human immunodeficiency virus type 1 Tat protein | Protein Tat | TAT_HV112 | Transactivating regulatory protein | tat
Type:PROTEIN
Mol. Mass.:9771.75
Organism:Human immunodeficiency virus type 1 (isolate PCV12 group M subtype B)(HIV-1)
Description:ChEMBL_199318
Residue:86
Sequence:
MEPVDPRLEPWKHPGSQPKTACTNCYCKKCCFHCQVCFITKALGISYGRKKRRQRRRAPQ
GSQTHQVSLSKQPTSQSRGDPTGPKE
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50097336
n/a
NameBDBM50097336
Synonyms:CHEMBL152397 | Pyrene-1-carboxylic acid [(4R,5S,6S)-5-amino-6-((2R,3R,4R)-4,6-diamino-2,3-dihydroxy-cyclohexyloxy)-3,4-dihydroxy-tetrahydro-pyran-2-ylmethyl]-amide
TypeSmall organic molecule
Emp. Form.C29H34N4O7
Mol. Mass.550.6029
SMILESNC1CC(N)C(OC2OC(CNC(=O)c3ccc4ccc5cccc6ccc3c4c56)C(O)C(O)C2N)C(O)C1O
Structure
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