Reaction Details |
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Target | Protein Tat |
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Ligand | BDBM50097336 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_209907 (CHEMBL811911) |
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Kd | 290±n/a nM |
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Citation | Hamasaki, K; Ueno, A Aminoglycoside antibiotics, neamine and its derivatives as potent inhibitors for the RNA-protein interactions derived from HIV-1 activators. Bioorg Med Chem Lett11:591-4 (2001) [PubMed] |
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More Info.: | Get all data from this article, Assay Method |
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Protein Tat |
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Name: | Protein Tat |
Synonyms: | Human immunodeficiency virus type 1 Tat protein | Protein Tat | TAT_HV112 | Transactivating regulatory protein | tat |
Type: | PROTEIN |
Mol. Mass.: | 9771.75 |
Organism: | Human immunodeficiency virus type 1 (isolate PCV12 group M subtype B)(HIV-1) |
Description: | ChEMBL_199318 |
Residue: | 86 |
Sequence: | MEPVDPRLEPWKHPGSQPKTACTNCYCKKCCFHCQVCFITKALGISYGRKKRRQRRRAPQ
GSQTHQVSLSKQPTSQSRGDPTGPKE
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BDBM50097336 |
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n/a |
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Name | BDBM50097336 |
Synonyms: | CHEMBL152397 | Pyrene-1-carboxylic acid [(4R,5S,6S)-5-amino-6-((2R,3R,4R)-4,6-diamino-2,3-dihydroxy-cyclohexyloxy)-3,4-dihydroxy-tetrahydro-pyran-2-ylmethyl]-amide |
Type | Small organic molecule |
Emp. Form. | C29H34N4O7 |
Mol. Mass. | 550.6029 |
SMILES | NC1CC(N)C(OC2OC(CNC(=O)c3ccc4ccc5cccc6ccc3c4c56)C(O)C(O)C2N)C(O)C1O |
Structure |
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