| Reaction Details |
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 | Report a problem with these data |
| Target | Melanocyte-stimulating hormone receptor |
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| Ligand | BDBM50111183 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_105842 |
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| Ki | 1300±n/a nM |
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| Citation |  Mutulis, F; Mutule, I; Wikberg, JE N-alkylaminoacids and their derivatives interact with melanocortin receptors. Bioorg Med Chem Lett12:1039-42 (2002) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Melanocyte-stimulating hormone receptor |
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| Name: | Melanocyte-stimulating hormone receptor |
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| Synonyms: | MC1-R | MC1R | MSH-R | MSHR | MSHR_HUMAN | Melanocortin MC1 | Melanocortin receptor (M1 and M4) | Melanocortin receptor 1 (MC-1) | Melanocortin receptor 1 (MC1-R) | Melanocortin receptor 1 (MC1R) |
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| Type: | Enzyme |
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| Mol. Mass.: | 34717.23 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q01726 |
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| Residue: | 317 |
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| Sequence: | MAVQGSQRRLLGSLNSTPTAIPQLGLAANQTGARCLEVSISDGLFLSLGLVSLVENALVV
ATIAKNRNLHSPMYCFICCLALSDLLVSGSNVLETAVILLLEAGALVARAAVLQQLDNVI
DVITCSSMLSSLCFLGAIAVDRYISIFYALRYHSIVTLPRARRAVAAIWVASVVFSTLFI
AYYDHVAVLLCLVVFFLAMLVLMAVLYVHMLARACQHAQGIARLHKRQRPVHQGFGLKGA
VTLTILLGIFFLCWGPFFLHLTLIVLCPEHPTCGCIFKNFNLFLALIICNAIIDPLIYAF
HSQELRRTLKEVLTCSW
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| BDBM50111183 |
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| n/a |
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| Name | BDBM50111183 |
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| Synonyms: | (2S)-5-[(E)-[amino(azaniumyl)methylidene]amino]-N-(naphthalen-1-yl)-2-[(naphthalen-2-ylmethyl)amino]pentanamide | MK-54 | N-Alkylaminoacid derivative |
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| Type | Small organic molecule |
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| Emp. Form. | C27H30N5O |
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| Mol. Mass. | 440.5595 |
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| SMILES | [NH3+]C(=N)NCCC[C@H](NCc1ccc2ccccc2c1)C(=O)Nc1cccc2ccccc12 |
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| Structure | 
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