| Reaction Details |
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 | Report a problem with these data |
| Target | Coagulation factor X |
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| Ligand | BDBM50118798 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_69660 (CHEMBL681852) |
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| Kd | 3500±n/a nM |
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| Citation |  Gunnarsson, GT; Desai, UR Exploring new non-sugar sulfated molecules as activators of antithrombin. Bioorg Med Chem Lett13:679-83 (2003) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Coagulation factor X |
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| Name: | Coagulation factor X |
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| Synonyms: | Activated coagulation factor X (FXa) | Activated factor Xa heavy chain | Coagulation factor X precursor | Coagulation factor Xa | F10 | FA10_HUMAN | Factor X heavy chain | Factor X light chain | Factor Xa | Stuart factor | Stuart-Prower factor |
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| Type: | Enzyme |
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| Mol. Mass.: | 54726.60 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 488 |
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| Sequence: | MGRPLHLVLLSASLAGLLLLGESLFIRREQANNILARVTRANSFLEEMKKGHLERECMEE
TCSYEEAREVFEDSDKTNEFWNKYKDGDQCETSPCQNQGKCKDGLGEYTCTCLEGFEGKN
CELFTRKLCSLDNGDCDQFCHEEQNSVVCSCARGYTLADNGKACIPTGPYPCGKQTLERR
KRSVAQATSSSGEAPDSITWKPYDAADLDPTENPFDLLDFNQTQPERGDNNLTRIVGGQE
CKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGE
AVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGI
VSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSG
GPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKTRGLPKAKSHAPE
VITSSPLK
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| BDBM50118798 |
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| n/a |
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| Name | BDBM50118798 |
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| Synonyms: | (+/-)-CS Sulfuric acid mono-[2-(3,4-bis-sulfooxy -phenyl)-3,5-bis-sulfooxy-chroman-7-yl] ester | (2S,3R)-2-[3,4-bis(sulfonatooxy)phenyl]-3,5-bis(sulfonatooxy)-3,4-dihydro-2H-chromen-7-yl sulfate |
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| Type | Small organic molecule |
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| Emp. Form. | C15H9O21S5 |
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| Mol. Mass. | 685.547 |
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| SMILES | [O-]S(=O)(=O)O[C@@H]1Cc2c(OS([O-])(=O)=O)cc(OS([O-])(=O)=O)cc2O[C@H]1c1ccc(OS([O-])(=O)=O)c(OS([O-])(=O)=O)c1 |
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| Structure | 
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