| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A2a |
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| Ligand | BDBM82015 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_75662 |
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| Ki | 400±n/a nM |
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| Citation |  Daly, JW Adenosine receptors: targets for future drugs. J Med Chem25:197-207 (1982) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A2a |
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| Name: | Adenosine receptor A2a |
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| Synonyms: | AA2AR_CAVPO | ADENOSINE A2 | ADORA2A | Adenosine A2a receptor |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 44955.08 |
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| Organism: | GUINEA PIG |
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| Description: | ADENOSINE A2 0 GUINEA PIG::P46616 |
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| Residue: | 409 |
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| Sequence: | MSSSVYITVELVIAVLAILGNVLVCWAVWINSNLQNVTNYFVVSLAAADIAVGVLAIPFA
ITISTGFCAACHGCLFFACFVLVLTQSSIFSLLTITIDRYIAIRIPLRYNGLVTCTRAKG
IIAICWVLSFAIGLTPMLGWNNCSQPKGDKNHSESCDEGQVTCLFEDVVPMNYMVYYNFF
AFVLVPLLLMLGIYLRIFLAARRQLKQMESQPLPGERTRSTLQKEVHPAKSLAIIVGLFA
LCCLPLNIINCFTFFCPECDHAPPWLMYLTIILSHGNSVVNPLIYAYRIREFRQTFRKII
RSHILRRRELFKAGGTSARASAAHSPEGEQVSLRLNGHPPGVWANGSALRPEQRPNGYVL
GLVSGRSAQRSHGDASLSDVELLSHEHKGTCPESPSLEDPPAHGGAGVS
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| BDBM82015 |
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| n/a |
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| Name | BDBM82015 |
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| Synonyms: | 1,3-Dimethyl-8-phenyl-3,9-dihydro-purine-2,6-dione | 8-Phenyltheophylline | CAS_1922 | CHEMBL62350 | NSC_1922 |
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| Type | Small organic molecule |
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| Emp. Form. | C13H12N4O2 |
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| Mol. Mass. | 256.26 |
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| SMILES | Cn1c2nc([nH]c2c(=O)n(C)c1=O)-c1ccccc1 |
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| Structure | 
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