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TargetAminopeptidase B
LigandBDBM50022742
Substrate/Competitorn/a
Meas. Tech.ChEBML_35352
Ki>1000000±n/a nM
Citation Ocain, TDRich, DH Synthesis of sulfur-containing analogues of bestatin. Inhibition of aminopeptidases by alpha-thiolbestatin analogues. J Med Chem31:2193-9 (1988) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Aminopeptidase B
Name:Aminopeptidase B
Synonyms:AMPB_RAT | Ap-B | Arginine aminopeptidase | Arginyl aminopeptidase | Cytosol aminopeptidase IV | Rnpep
Type:PROTEIN
Mol. Mass.:72609.93
Organism:Rattus norvegicus
Description:ChEMBL_1344423
Residue:650
Sequence:
MESSGPSSCHSAARRPLHSAQAVDVASASSFRAFEILHLHLDLRAEFGPPGPGPGSRGLN
GKATLELRCLLPEGASELRLDSHSCLEVMAATLLRGQPGDQQQLTEPVPFHTQPFSHYGQ
ALCVVFPKPCCAAERFRLELTYRVGEGPGVCWLAPEQTAGKKKPFVYTQGQAVLNRAFFP
CFDTPAVKCTYSALVEVPDGFTAVMSASTWERRGPNKFFFQMSQPIPSYLIALAIGDLAS
AEVGPRSRVWAEPCLIEAAKEEYNGVIEEFLATGEKLFGPYVWGRYDLLFMPPSFPFGGM
ENPCLTFVTPCLLAGDRSLADVIIHEISHSWFGNLVTNANWGEFWLNEGFTMYAQRRIST
ILFGAAYTCLEAATGRALLRQHMDVSGEENPLNKLRVKIEPGVDPDDTYNETPYEKGYCF
VSYLAHLVGDQEQFDKFLKAYVDEFKFQSILAEDFLEFYLEYFPELKKKGVDSIPGFEFN
RWLNTPGWPPYLPDLSPGDSLMKPAEELAELWAASEPDMQAIEAVAISTWKTYQLVYFLD
KILQKSPLPPGNVKKLGETYPKISNAQNAELRLRWGQIILKNDHQEEFWKVKDFLQSQGK
QKYTLPLYHAMMGGSEMARTLAKETFSATASQLHSNVVNYVQQILAPKGS
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50022742
n/a
NameBDBM50022742
Synonyms:3-Amino-2-hydroxy-N-(3-methyl-butyl)-4-phenyl-thiobutyramide; Trifluoro acetate | CHEMBL67868
TypeSmall organic molecule
Emp. Form.C15H24N2OS
Mol. Mass.280.429
SMILESCC(C)CCNC(=S)[C@@H](O)[C@H](N)Cc1ccccc1
Structure
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