| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Indolethylamine N-methyltransferase |
|---|
| Ligand | BDBM50367839 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEBML_89038 |
|---|
| Ki | 12000±n/a nM |
|---|
| Citation |  Broom, AD Rational design of enzyme inhibitors: multisubstrate analogue inhibitors. J Med Chem32:2-7 (1989) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Indolethylamine N-methyltransferase |
|---|
| Name: | Indolethylamine N-methyltransferase |
|---|
| Synonyms: | Amine N-methyltransferase | Aromatic alkylamine N-methyltransferase | Arylamine N-methyltransferase | INMT | INMT_HUMAN | Indolamine N-methyltransferase |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 28884.19 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_1333668 |
|---|
| Residue: | 263 |
|---|
| Sequence: | MKGGFTGGDEYQKHFLPRDYLATYYSFDGSPSPEAEMLKFNLECLHKTFGPGGLQGDTLI
DIGSGPTIYQVLAACDSFQDITLSDFTDRNREELEKWLKKEPGAYDWTPAVKFACELEGN
SGRWEEKEEKLRAAVKRVLKCDVHLGNPLAPAVLPLADCVLTLLAMECACCSLDAYRAAL
CNLASLLKPGGHLVTTVTLRLPSYMVGKREFSCVALEKEEVEQAVLDAGFDIEQLLHSPQ
SYSVTNAANNGVCFIVARKKPGP
|
|
|
|---|
| BDBM50367839 |
|---|
| n/a |
|---|
| Name | BDBM50367839 |
|---|
| Synonyms: | CHEMBL2368635 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C23H29IN6O3S |
|---|
| Mol. Mass. | 596.484 |
|---|
| SMILES | [I-].C[S+](CCCCc1c[nH]c2ccccc12)C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12 |r| |
|---|
| Structure | 
|
|---|
Search and Browse
