| Reaction Details |
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 | Report a problem with these data |
| Target | D(1A) dopamine receptor |
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| Ligand | BDBM50010291 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_60185 (CHEMBL872877) |
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| Ki | 10000±n/a nM |
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| Citation |  Bakthavachalam, V; Baindur, N; Madras, BK; Neumeyer, JL Fluorescent probes for dopamine receptors: synthesis and characterization of fluorescein and 7-nitrobenz-2-oxa-1,3-diazol-4-yl conjugates of D-1 and D-2 receptor ligands. J Med Chem34:3235-41 (1991) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| D(1A) dopamine receptor |
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| Name: | D(1A) dopamine receptor |
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| Synonyms: | DA D1 receptor | DOPAMINE D1 | DRD1 | DRD1_HUMAN | Dopamine D1 receptor | Dopamine D1 receptor (D1R) | Dopamine D1A |
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| Type: | Enzyme |
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| Mol. Mass.: | 49303.43 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21728 |
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| Residue: | 446 |
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| Sequence: | MRTLNTSAMDGTGLVVERDFSVRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTN
FFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVD
RYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTSPSDGNATSLA
ETIDNCDSSLSRTYAISSSVISFYIPVAIMIVTYTRIYRIAQKQIRRIAALERAAVHAKN
CQTTTGNGKPVECSQPESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFILNCILPFCGS
GETQPFCIDSNTFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCYRLCPATNNAIET
VSINNNGAAMFSSHHEPRGSISKECNLVYLIPHAVGSSEDLKKEEAAGIARPLEKLSPAL
SVILDYDTDVSLEKIQPITQNGQHPT
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| BDBM50010291 |
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| n/a |
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| Name | BDBM50010291 |
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| Synonyms: | 5-[4-(7,8-dihydroxy-2,3,4,5-tetrahydro-1H-benzo[d]azepin-1-yl)anilino(thioxo)methylamino]-3',6'-dihydroxyspiro[1,3-dihydroisobenzofuran-1,9'-(9'H-xanthene)]-3-onehydrochloride | CHEMBL538023 |
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| Type | Small organic molecule |
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| Emp. Form. | C37H29N3O7S |
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| Mol. Mass. | 659.707 |
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| SMILES | Oc1ccc2c(Oc3cc(O)ccc3C22OC(=O)c3cc(NC(=S)Nc4ccc(cc4)C4CNCCc5cc(O)c(O)cc45)ccc23)c1 |
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| Structure | 
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