| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50036138 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_145429 (CHEMBL748774) |
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| Ki | 136±n/a nM |
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| Citation |  Portoghese, PS; Farouz-Grant, F; Sultana, M; Takemori, AE 7'-Substituted amino acid conjugates of naltrindole. Hydrophilic groups as determinants of selective antagonism of delta 1 opioid receptor-mediated antinociception in mice. J Med Chem38:402-7 (1995) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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| BDBM50036138 |
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| n/a |
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| Name | BDBM50036138 |
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| Synonyms: | 5-amino-2-[22-cyclopropylmethyl-2,16-dihydroxy-(2S,13R)-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaen-9-ylcarboxamido]-(2R)-pentanoic acid | CHEMBL132897 |
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| Type | Small organic molecule |
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| Emp. Form. | C32H36N4O6 |
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| Mol. Mass. | 572.6514 |
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| SMILES | NCCC[C@@H](NC(=O)c1cccc2c3C[C@@]4(O)C5Cc6ccc(O)c7O[C@@H](c3[nH]c12)C4(CCN5CC1CC1)c67)C(O)=O |TLB:34:33:15:38.19.18,24:38:15:33.31.32,16:15:38.19.18:33.31.32,THB:14:15:38.19.18:33.31.32| |
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| Structure | 
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