| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50254511 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_147110 (CHEMBL758273) |
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| IC50 | 1.1±n/a nM |
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| Citation |  Davis, RD; Nelson, WL Isothiocyanate-substituted benzyl ether opioid receptor ligands derived from 6 beta-naltrexol. J Med Chem38:570-9 (1995) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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|
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| BDBM50254511 |
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| n/a |
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| Name | BDBM50254511 |
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| Synonyms: | CHEMBL468469 | Naltrexone-6-alpha-ol |
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| Type | Small organic molecule |
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| Emp. Form. | C20H25NO4 |
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| Mol. Mass. | 343.4168 |
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| SMILES | O[C@H]1CC[C@@]2(O)[C@H]3Cc4ccc(O)c5O[C@@H]1[C@]2(CCN3CC1CC1)c45 |r| |
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| Structure | 
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