Reaction Details |
| Report a problem with these data |
Target | Muscarinic receptor M1 |
---|
Ligand | BDBM50055978 |
---|
Substrate/Competitor | n/a |
---|
Meas. Tech. | ChEMBL_140161 (CHEMBL745466) |
---|
Ki | 0.02±n/a nM |
---|
Citation | Visser, TJ; van Waarde, A; Jansen, TJ; Visser, GM; van der Mark, TW; Kraan, J; Ensing, K; Vaalburg, W Stereoselective synthesis and biodistribution of potent [11C]-labeled antagonists for positron emission tomography imaging of muscarinic receptors in the airways. J Med Chem40:117-24 (1997) [PubMed] Article |
---|
More Info.: | Get all data from this article, Assay Method |
---|
|
Muscarinic receptor M1 |
---|
Name: | Muscarinic receptor M1 |
Synonyms: | Muscarinic acetylcholine receptor M1 |
Type: | PROTEIN |
Mol. Mass.: | 15022.43 |
Organism: | Bos taurus |
Description: | ChEMBL_140161 |
Residue: | 139 |
Sequence: | ETENRARELAALQGSETPGKGGGSSSSSERSQPGAEGSPETPPGRCCRCCRTPRLLQAYS
WKEEEEEDEGSMESLTSSEGEEPGSEVVIKMPMVDPEAQAPAKQPPRSSPNTVKRPTRKG
RERAGKGQKPRGKEQLAKR
|
|
|
BDBM50055978 |
---|
n/a |
---|
Name | BDBM50055978 |
Synonyms: | 4-((R)-2-Cyclohexyl-2-hydroxy-2-phenyl-acetoxy)-1,1-dimethyl-piperidinium; iodide | CHEMBL21905 |
Type | Small organic molecule |
Emp. Form. | C21H32NO3 |
Mol. Mass. | 346.4831 |
SMILES | C[N+]1(C)CCC(CC1)OC(=O)[C@@](O)(C1CCCCC1)c1ccccc1 |
Structure |
|