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TargetMuscarinic receptor M1
LigandBDBM50055978
Substrate/Competitorn/a
Meas. Tech.ChEMBL_140161 (CHEMBL745466)
Ki 0.02±n/a nM
Citation Visser, TJvan Waarde, AJansen, TJVisser, GMvan der Mark, TWKraan, JEnsing, KVaalburg, W Stereoselective synthesis and biodistribution of potent [11C]-labeled antagonists for positron emission tomography imaging of muscarinic receptors in the airways. J Med Chem40:117-24 (1997) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Muscarinic receptor M1
Name:Muscarinic receptor M1
Synonyms:Muscarinic acetylcholine receptor M1
Type:PROTEIN
Mol. Mass.:15022.43
Organism:Bos taurus
Description:ChEMBL_140161
Residue:139
Sequence:
ETENRARELAALQGSETPGKGGGSSSSSERSQPGAEGSPETPPGRCCRCCRTPRLLQAYS
WKEEEEEDEGSMESLTSSEGEEPGSEVVIKMPMVDPEAQAPAKQPPRSSPNTVKRPTRKG
RERAGKGQKPRGKEQLAKR
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50055978
n/a
NameBDBM50055978
Synonyms:4-((R)-2-Cyclohexyl-2-hydroxy-2-phenyl-acetoxy)-1,1-dimethyl-piperidinium; iodide | CHEMBL21905
TypeSmall organic molecule
Emp. Form.C21H32NO3
Mol. Mass.346.4831
SMILESC[N+]1(C)CCC(CC1)OC(=O)[C@@](O)(C1CCCCC1)c1ccccc1
Structure
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