| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM50058659 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_146320 (CHEMBL757529) |
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| Ki | 0.41±n/a nM |
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| Citation |  Farouz-Grant, F; Portoghese, PS Pyrrolomorphinans as delta opioid receptor antagonists. The role of steric hindrance in conferring selectivity. J Med Chem40:1977-81 (1997) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40577.25 |
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| Organism: | MOUSE |
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| Description: | P32300 |
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| Residue: | 372 |
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| Sequence: | MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTAC
TPSDGPGGGAAA
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| BDBM50058659 |
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| n/a |
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| Name | BDBM50058659 |
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| Synonyms: | 18-cyclopropylmethyl-5,6-dimethyl-10-oxa-7,18-diazahexacyclo[9.9.1.01,9.02,17.04,8.015,21]henicosa-4(8),5,11,13,15(21)-pentaene-2,12-diol | CHEMBL60404 |
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| Type | Small organic molecule |
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| Emp. Form. | C24H28N2O3 |
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| Mol. Mass. | 392.4907 |
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| SMILES | Cc1[nH]c2[C@@H]3Oc4c5c(CC6N(CC7CC7)CCC35[C@@]6(O)Cc2c1C)ccc4O |THB:12:11:19:7.8.9,6:7:19:11.17.16,20:19:7.8.9:11.17.16| |
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| Structure | 
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