| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 2 |
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| Ligand | BDBM50059091 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_200501 (CHEMBL803846) |
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| IC50 | 13±n/a nM |
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| Citation |  Osapay, G; Prokai, L; Kim, HS; Medzihradszky, KF; Coy, DH; Liapakis, G; Reisine, T; Melacini, G; Zhu, Q; Wang, SH; Mattern, RH; Goodman, M Lanthionine-somatostatin analogs: synthesis, characterization, biological activity, and enzymatic stability studies. J Med Chem40:2241-51 (1997) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 2 |
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| Name: | Somatostatin receptor type 2 |
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| Synonyms: | SOMATOSTATIN SST2 | SSR2_MOUSE | Smstr2 | Somatostatin receptor | Somatostatin receptor 2 | Somatostatin receptor type 2 | Sst2 | Sstr2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 41234.26 |
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| Organism: | MOUSE |
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| Description: | SOMATOSTATIN SST2 SSTR2 MOUSE::P30875 |
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| Residue: | 369 |
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| Sequence: | MEMSSEQLNGSQVWVSSPFDLNGSLGPSNGSNQTEPYYDMTSNAVLTFIYFVVCVVGLCG
NTLVIYVILRYAKMKTITNIYILNLAIADELFMLGLPFLAMQVALVHWPFGKAICRVVMT
VDGINQFTSIFCLTVMSIDRYLAVVHPIKSAKWRRPRTAKMINVAVWCVSLLVILPIMIY
AGLRSNQWGRSSCTINWPGESGAWYTGFIIYAFILGFLVPLTIICLCYLFIIIKVKSSGI
RVGSSKRKKSEKKVTRMVSIVVAVFIFCWLPFYIFNVSSVSVAISPTPALKGMFDFVVIL
TYANSCANPILYAFLSDNFKKSFQNVLCLVKVSGTEDGERSDSKQDKSRLNETTETQRTL
LNGDLQTSI
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| BDBM50059091 |
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| n/a |
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| Name | BDBM50059091 |
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| Synonyms: | 2-{[9-(4-Amino-butyl)-18-(2-amino-3-phenyl-propionylamino)-15-benzyl-6-(1-hydroxy-ethyl)-12-(1H-indol-3-ylmethyl)-5,8,11,14,17-pentaoxo-1-thia-4,7,10,13,16-pentaaza-cyclononadecane-3-carbonyl]-amino}-3-hydroxy-butyric acid | CHEMBL266469 |
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| Type | Small organic molecule |
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| Emp. Form. | C49H64N10O11S |
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| Mol. Mass. | 1001.158 |
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| SMILES | C[C@@H](O)[C@H](NC(=O)[C@@H]1CSC[C@@H](NC(=O)[C@H](N)Cc2ccccc2)C(=O)N[C@H](Cc2ccccc2)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@H](CCCCN)C(=O)N[C@@H]([C@@H](C)O)C(=O)N1)C(O)=O |
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| Structure | 
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