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TargetMu-type opioid receptor
LigandBDBM50369588
Substrate/Competitorn/a
Meas. Tech.ChEMBL_145274 (CHEMBL751210)
Ki 240±n/a nM
Citation Wentland, MPDuan, WCohen, DJBidlack, JM Selective protection and functionalization of morphine: synthesis and opioid receptor binding properties of 3-amino-3-desoxymorphine derivatives. J Med Chem43:3558-65 (2000) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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  Blast E-value cutoff:
BDBM50369588
n/a
NameBDBM50369588
Synonyms:CHEMBL119332
TypeSmall organic molecule
Emp. Form.C19H24N2O2
Mol. Mass.312.4061
SMILESCN(C)c1ccc2C[C@@H]3[C@@H]4C=C[C@H](O)[C@@H]5Oc1c2[C@]45CCN3C |c:10|
Structure
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