| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50092176 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_145274 (CHEMBL751210) |
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| Ki | 1.8±n/a nM |
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| Citation |  Wentland, MP; Duan, W; Cohen, DJ; Bidlack, JM Selective protection and functionalization of morphine: synthesis and opioid receptor binding properties of 3-amino-3-desoxymorphine derivatives. J Med Chem43:3558-65 (2000) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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|
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| BDBM50092176 |
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| n/a |
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| Name | BDBM50092176 |
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| Synonyms: | 3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ylamine | CHEMBL332017 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H26N2 |
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| Mol. Mass. | 270.4124 |
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| SMILES | C[C@H]1[C@H]2Cc3ccc(N)cc3[C@@]1(C)CCN2CC1CC1 |TLB:16:15:1:10.4.3| |
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| Structure | 
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