| Reaction Details |
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 | Report a problem with these data |
| Target | P2Y purinoceptor 1 |
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| Ligand | BDBM50085827 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_147720 (CHEMBL759190) |
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| EC50 | 41000±n/a nM |
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| Citation |  Nandanan, E; Jang, SY; Moro, S; Kim, HO; Siddiqui, MA; Russ, P; Marquez, VE; Busson, R; Herdewijn, P; Harden, TK; Boyer, JL; Jacobson, KA Synthesis, biological activity, and molecular modeling of ribose-modified deoxyadenosine bisphosphate analogues as P2Y(1) receptor ligands. J Med Chem43:829-42 (2000) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| P2Y purinoceptor 1 |
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| Name: | P2Y purinoceptor 1 |
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| Synonyms: | P2RY1 | P2RY1_MELGA |
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| Type: | n/a |
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| Mol. Mass.: | 41199.64 |
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| Organism: | Meleagris gallopavo |
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| Description: | n/a |
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| Residue: | 362 |
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| Sequence: | MTEALISAALNGTQPELLAGGWAAGNASTKCSLTKTGFQFYYLPTVYILVFITGFLGNSV
AIWMFVFHMRPWSGISVYMFNLALADFLYVLTLPALIFYYFNKTDWIFGDVMCKLQRFIF
HVNLYGSILFLTCISVHRYTGVVHPLKSLGRLKKKNAVYVSSLVWALVVAVIAPILFYSG
TGVRRNKTITCYDTTADEYLRSYFVYSMCTTVFMFCIPFIVILGCYGLIVKALIYKDLDN
SPLRRKSIYLVIIVLTVFAVSYLPFHVMKTLNLRARLDFQTPQMCAFNDKVYATYQVTRG
LASLNSCVDPILYFLAGDTFRRRLSRATRKSSRRSEPNVQSKSEEMTLNILTEYKQNGDT
SL
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| BDBM50085827 |
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| n/a |
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| Name | BDBM50085827 |
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| Synonyms: | CHEMBL169580 | Phosphoric acid mono-[5-(6-methylamino-purin-9-yl)-3-phosphonooxy-tetrahydro-furan-2-yl] ester |
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| Type | Small organic molecule |
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| Emp. Form. | C12H22N6O14P4 |
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| Mol. Mass. | 598.2299 |
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| SMILES | Nc1ncnc2n(cnc12)C1CN(CCP(O)(O)=O)CC(COP(O)(=O)OP(O)(=O)OP(O)(O)=O)O1 |
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| Structure | 
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