| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Somatostatin receptor type 1 |
|---|
| Ligand | BDBM50369890 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_200666 (CHEMBL806158) |
|---|
| Ki | >10000±n/a nM |
|---|
| Citation |  Poitout, L; Roubert, P; Contour-Galcéra, MO; Moinet, C; Lannoy, J; Pommier, J; Plas, P; Bigg, D; Thurieau, C Identification of potent non-peptide somatostatin antagonists with sst(3) selectivity. J Med Chem44:2990-3000 (2001) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Somatostatin receptor type 1 |
|---|
| Name: | Somatostatin receptor type 1 |
|---|
| Synonyms: | SOMATOSTATIN SST1 | SRIF-2 | SS-1-R | SS1-R | SS1R | SSR1_HUMAN | SSTR1 | Somatostatin receptor type 1 (SSTR1) |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 42692.81 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P30872 |
|---|
| Residue: | 391 |
|---|
| Sequence: | MFPNGTASSPSSSPSPSPGSCGEGGGSRGPGAGAADGMEEPGRNASQNGTLSEGQGSAIL
ISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLL
RHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLG
VWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAIC
LCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQD
DATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKS
RAYSVEDFQPENLESGGVFRNGTCTSRITTL
|
|
|
|---|
| BDBM50369890 |
|---|
| n/a |
|---|
| Name | BDBM50369890 |
|---|
| Synonyms: | CHEMBL1237140 | CHEMBL1788167 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C28H34N4 |
|---|
| Mol. Mass. | 426.5964 |
|---|
| SMILES | CCCCC1(CCCC)N[C@@H](Cc2c1[nH]c1ccccc21)c1nc(c[nH]1)-c1ccccc1 |r| |
|---|
| Structure | 
|
|---|
Search and Browse
