| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM50107597 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_46986 (CHEMBL658955) |
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| Ki | 70±n/a nM |
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| Citation |  López-Rodríguez, ML; Viso, A; Ortega-Gutiérrez, S; Lastres-Becker, I; González, S; Fernández-Ruiz, J; Ramos, JA Design, synthesis and biological evaluation of novel arachidonic acid derivatives as highly potent and selective endocannabinoid transporter inhibitors. J Med Chem44:4505-8 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 39690.94 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P34972 |
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| Residue: | 360 |
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| Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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| BDBM50107597 |
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| n/a |
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| Name | BDBM50107597 |
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| Synonyms: | (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid (1-methyl-1H-pyrrol-2-ylmethyl)-amide | CHEMBL417158 | Icosa-5,8,11,14-tetraenoic acid (1-methyl-1H-pyrrol-2-ylmethyl)-amide |
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| Type | Small organic molecule |
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| Emp. Form. | C26H40N2O |
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| Mol. Mass. | 396.6086 |
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| SMILES | CCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCC(=O)NCc1cccn1C |
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| Structure | 
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