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TargetAdenosine receptor A1
LigandBDBM50369987
Substrate/Competitorn/a
Meas. Tech.ChEMBL_29318
Ki 38.10±n/a nM
Citation Rieger JMBrown MLSullivan GWLinden JMacdonald TL Design, synthesis, and evaluation of novel A2A adenosine receptor agonists. J Med Chem 44:531-9 (2001) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Adenosine receptor A1
Name:Adenosine receptor
Synonyms:ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | Adenosine A1 receptor (A1) | Adenosine receptors A1
Type:Protein
Mol. Mass.:36704.13
Organism:Rattus norvegicus (rat)
Description:n/a
Residue:326
Sequence:
MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVT
QRRAAVAIAGCWILSLVVGLTPMFGWNNLSVVEQDWRANGSVGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALIL
FLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFL
KIWNDHFRCQPKPPIDEDLPEEKAED
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  Blast E-value cutoff:
BDBM50369987
n/a
NameBDBM50369987
Synonyms:CHEMBL608460
TypeSmall organic molecule
Emp. Form.C12H17N5O5
Mol. Mass.311.2939
SMILESCOCc1nc(N)c2ncn(C3O[C@H](CO)[C@@H](O)[C@H]3O)c2n1 |r|
Structure
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