| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 1 |
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| Ligand | BDBM50370052 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_200541 (CHEMBL805045) |
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| Ki | 1000±n/a nM |
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| Citation |  Rajeswaran, WG; Hocart, SJ; Murphy, WA; Taylor, JE; Coy, DH Highly potent and subtype selective ligands derived by N-methyl scan of a somatostatin antagonist. J Med Chem44:1305-11 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 1 |
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| Name: | Somatostatin receptor type 1 |
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| Synonyms: | SOMATOSTATIN SST1 | SRIF-2 | SS-1-R | SS1-R | SS1R | SSR1_HUMAN | SSTR1 | Somatostatin receptor type 1 (SSTR1) |
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| Type: | Enzyme |
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| Mol. Mass.: | 42692.81 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P30872 |
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| Residue: | 391 |
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| Sequence: | MFPNGTASSPSSSPSPSPGSCGEGGGSRGPGAGAADGMEEPGRNASQNGTLSEGQGSAIL
ISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLL
RHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLG
VWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAIC
LCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQD
DATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKS
RAYSVEDFQPENLESGGVFRNGTCTSRITTL
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| BDBM50370052 |
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| n/a |
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| Name | BDBM50370052 |
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| Synonyms: | CHEMBL1794046 |
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| Type | Small organic molecule |
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| Emp. Form. | C61H73ClN12O9S2 |
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| Mol. Mass. | 1217.89 |
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| SMILES | CNC(=O)C(NC(=O)[C@H]1CSSC[C@H](N(C)C(=O)C(N)Cc2ccc(Cl)cc2)C(=O)NC(Cc2cccnc2)C(=O)N[C@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CCCCN)C(=O)N[C@H]([C@H](C)O)C(=O)N1)C(c1ccccc1)c1ccccc1 |
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| Structure | 
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