| Reaction Details |
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 | Report a problem with these data |
| Target | P2X purinoceptor 4 |
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| Ligand | BDBM50118234 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_149737 (CHEMBL759520) |
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| IC50 | 9600±n/a nM |
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| Citation |  Jacobson, KA; Jarvis, MF; Williams, M Purine and pyrimidine (P2) receptors as drug targets. J Med Chem45:4057-93 (2002) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| P2X purinoceptor 4 |
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| Name: | P2X purinoceptor 4 |
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| Synonyms: | P2RX4_RAT | P2rx4 | Purinergic, P2X4 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 43504.16 |
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| Organism: | RAT |
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| Description: | Purinergic, P2X4 0 RAT::P51577 |
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| Residue: | 388 |
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| Sequence: | MAGCCSVLGSFLFEYDTPRIVLIRSRKVGLMNRAVQLLILAYVIGWVFVWEKGYQETDSV
VSSVTTKAKGVAVTNTSQLGFRIWDVADYVIPAQEENSLFIMTNMIVTVNQTQSTCPEIP
DKTSICNSDADCTPGSVDTHSSGVATGRCVPFNESVKTCEVAAWCPVENDVGVPTPAFLK
AAENFTLLVKNNIWYPKFNFSKRNILPNITTSYLKSCIYNAQTDPFCPIFRLGTIVEDAG
HSFQEMAVEGGIMGIQIKWDCNLDRAASLCLPRYSFRRLDTRDLEHNVSPGYNFRFAKYY
RDLAGKEQRTLTKAYGIRFDIIVFGKAGKFDIIPTMINVGSGLALLGVATVLCDVIVLYC
MKKKYYYRDKKYKYVEDYEQGLSGEMNQ
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| BDBM50118234 |
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| n/a |
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| Name | BDBM50118234 |
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| Synonyms: | CHEMBL129904 | MRS 2160 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H13ClN3O8P |
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| Mol. Mass. | 429.706 |
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| SMILES | Cc1nc(N=Nc2ccc(C(O)=O)c(Cl)c2)c(COP(O)(O)=O)c(C=O)c1O |w:5.5| |
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| Structure | 
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