| Reaction Details |
|---|
 | Report a problem with these data |
| Target | P2Y purinoceptor 1 |
|---|
| Ligand | BDBM50118234 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_147575 (CHEMBL751772) |
|---|
| Kd | 2900±n/a nM |
|---|
| Citation |  Jacobson, KA; Jarvis, MF; Williams, M Purine and pyrimidine (P2) receptors as drug targets. J Med Chem45:4057-93 (2002) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| P2Y purinoceptor 1 |
|---|
| Name: | P2Y purinoceptor 1 |
|---|
| Synonyms: | ATP receptor | P2RY1 | P2RY1_HUMAN | P2Y purinoceptor 1 (P2Y1) | P2Y1 | Purinergic receptor | Purinergic receptor P2Y1 |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 42090.25 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P47900 |
|---|
| Residue: | 373 |
|---|
| Sequence: | MTEVLWPAVPNGTDAAFLAGPGSSWGNSTVASTAAVSSSFKCALTKTGFQFYYLPAVYIL
VFIIGFLGNSVAIWMFVFHMKPWSGISVYMFNLALADFLYVLTLPALIFYYFNKTDWIFG
DAMCKLQRFIFHVNLYGSILFLTCISAHRYSGVVYPLKSLGRLKKKNAICISVLVWLIVV
VAISPILFYSGTGVRKNKTITCYDTTSDEYLRSYFIYSMCTTVAMFCVPLVLILGCYGLI
VRALIYKDLDNSPLRRKSIYLVIIVLTVFAVSYIPFHVMKTMNLRARLDFQTPAMCAFND
RVYATYQVTRGLASLNSCVDPILYFLAGDTFRRRLSRATRKASRRSEANLQSKSEDMTLN
ILPEFKQNGDTSL
|
|
|
|---|
| BDBM50118234 |
|---|
| n/a |
|---|
| Name | BDBM50118234 |
|---|
| Synonyms: | CHEMBL129904 | MRS 2160 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C15H13ClN3O8P |
|---|
| Mol. Mass. | 429.706 |
|---|
| SMILES | Cc1nc(N=Nc2ccc(C(O)=O)c(Cl)c2)c(COP(O)(O)=O)c(C=O)c1O |w:5.5| |
|---|
| Structure | 
|
|---|
Search and Browse
