| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 1 |
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| Ligand | BDBM50103430 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_200542 (CHEMBL805046) |
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| Ki | 2392±n/a nM |
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| Citation |  Patchett, AA 2002 Alfred Burger Award Address in Medicinal Chemistry. Natural products and design: interrelated approaches in drug discovery. J Med Chem45:5609-16 (2002) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 1 |
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| Name: | Somatostatin receptor type 1 |
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| Synonyms: | SOMATOSTATIN SST1 | SRIF-2 | SS-1-R | SS1-R | SS1R | SSR1_HUMAN | SSTR1 | Somatostatin receptor type 1 (SSTR1) |
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| Type: | Enzyme |
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| Mol. Mass.: | 42692.81 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P30872 |
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| Residue: | 391 |
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| Sequence: | MFPNGTASSPSSSPSPSPGSCGEGGGSRGPGAGAADGMEEPGRNASQNGTLSEGQGSAIL
ISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLL
RHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLG
VWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAIC
LCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQD
DATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKS
RAYSVEDFQPENLESGGVFRNGTCTSRITTL
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| BDBM50103430 |
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| n/a |
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| Name | BDBM50103430 |
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| Synonyms: | 6-Amino-2-(3-(1H-indol-3-yl)-2-{[4-(2-oxo-2,3-dihydro-benzoimidazol-1-yl)-piperidine-1-carbonyl]-amino}-butyrylamino)-hexanoic acid tert-butyl ester | CHEMBL99895 |
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| Type | Small organic molecule |
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| Emp. Form. | C35H47N7O5 |
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| Mol. Mass. | 645.7916 |
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| SMILES | C[C@H]([C@@H](NC(=O)N1CCC(CC1)n1c2ccccc2[nH]c1=O)C(=O)N[C@@H](CCCCN)C(=O)OC(C)(C)C)c1c[nH]c2ccccc12 |
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| Structure | 
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