| Reaction Details |
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 | Report a problem with these data |
| Target | D(2) dopamine receptor |
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| Ligand | BDBM50122738 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_59634 (CHEMBL672424) |
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| Ki | 35400±n/a nM |
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| Citation |  Macchia, M; Cervetto, L; Demontis, GC; Longoni, B; Minutolo, F; Orlandini, E; Ortore, G; Papi, C; Sbrana, A; Macchia, B New N-n-propyl-substituted 3-aryl- and 3-cyclohexylpiperidines as partial agonists at the D4 dopamine receptor. J Med Chem46:161-8 (2002) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(2) dopamine receptor |
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| Name: | D(2) dopamine receptor |
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| Synonyms: | DOPAMINE D2 | DRD2 | DRD2_BOVIN | Dopamine D2 receptor |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 50698.79 |
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| Organism: | BOVINE |
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| Description: | P20288 |
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| Residue: | 444 |
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| Sequence: | MDPLNLSWYDDDPESRNWSRPFNGSEGKADRPPYNYYAMLLTLLIFVIVFGNVLVCMAVS
REKALQTTTNYLIVSLAVADLLVATLVMPWVVYLEVVGEWKFSRIHCDIFVTLDVMMCTA
SILNLCAISIDRYTAVAMPMLYNTRYSSKRRVTVMIAIVWVLSFTISCPMLFGLNNTDQN
ECIIANPAFVVYSSIVSFYVPFIVTLLVYIKIYIVLRRRRKRVNTKRSSRAFRANLKAPL
KGNCTHPEDMKLCTVIMKSNGSFPVNRRRVEAARRAQELEMEMLSSTSPPERTRYSPIPP
SHHQLTLPDPSHHGLHSTPDSPAKPEKNGHAKTVNPKIAKIFEIQSMPNGKTRTSLKTMS
RRKLSQQKEKKATQMLAIVLGVFIICWLPFFITHILNIHCDCNIPPVLYSAFTWLGYVNS
AVNPIIYTTFNIEFRKAFLKILHC
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| BDBM50122738 |
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| n/a |
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| Name | BDBM50122738 |
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| Synonyms: | 1-Propyl-3-p-tolyl-piperidine; hydrochloride | CHEMBL543078 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H23N |
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| Mol. Mass. | 217.3498 |
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| SMILES | CCCN1CCCC(C1)c1ccc(C)cc1 |
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| Structure | 
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