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TargetHydroxycarboxylic acid receptor 2
LigandBDBM50132135
Substrate/Competitorn/a
Meas. Tech.ChEMBL_144336
Ki>100000±n/a nM
Citation van Herk TBrussee Jvan den Nieuwendijk AMvan der Klein PAIJzerman APStannek CBurmeister ALorenzen A Pyrazole derivatives as partial agonists for the nicotinic acid receptor. J Med Chem 46:3945-51 (2003) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Hydroxycarboxylic acid receptor 2
Name:Hydroxycarboxylic acid receptor 2
Synonyms:HM74 nicotinic acid GPCR
Type:PROTEIN
Mol. Mass.:41476.06
Organism:Rattus norvegicus
Description:ChEMBL_820675
Residue:360
Sequence:
MSKQNHFLVINGKNCCVFRDENIAKVLPPVLGLEFVFGLLGNGLALWIFCFHLKSWKSSR
IFLFNLAVADFLLIICLPFLTDNYVQNWDWRFGSIPCRVMLFMLAMNRQGSIIFLTVVAV
DRYFRVVHPHHFLNKISNRTAAIISCFLWGITIGLTVHLLYTDMMTRNGDANLCSSFSIC
YTFRWHDAMFLLEFFLPLGIILFCSGRIIWSLRQRQMDRHVKIKRAINFIMVVAIVFVIC
FLPSVAVRIRIFWLLYKHNVRNCDIYSSVDLAFFTTLSFTYMNSMLDPVVYYFSSPSFPN
FFSTCINRCLRRKTLGEPDNNRSTSVELTGDPSTIRSIPGALMTDPSEPGSPPYLASTSR
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50132135
n/a
NameBDBM50132135
Synonyms:4,6-Dihydro-1H-furo[3,4-c]pyrazole-3-carboxylic acid | 4,6-dihydro-2H-furo[3,4-c]pyrazole-3-carboxylic acid | CHEMBL338071
TypeSmall organic molecule
Emp. Form.C6H6N2O3
Mol. Mass.154.1234
SMILESOC(=O)c1[nH]nc2COCc12
Structure
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