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TargetHydroxycarboxylic acid receptor 2
LigandBDBM50211363
Substrate/Competitorn/a
Meas. Tech.ChEMBL_144336
Ki 683±n/a nM
Citation van Herk TBrussee Jvan den Nieuwendijk AMvan der Klein PAIJzerman APStannek CBurmeister ALorenzen A Pyrazole derivatives as partial agonists for the nicotinic acid receptor. J Med Chem 46:3945-51 (2003) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Hydroxycarboxylic acid receptor 2
Name:Hydroxycarboxylic acid receptor 2
Synonyms:HM74 nicotinic acid GPCR
Type:PROTEIN
Mol. Mass.:41476.06
Organism:Rattus norvegicus
Description:ChEMBL_820675
Residue:360
Sequence:
MSKQNHFLVINGKNCCVFRDENIAKVLPPVLGLEFVFGLLGNGLALWIFCFHLKSWKSSR
IFLFNLAVADFLLIICLPFLTDNYVQNWDWRFGSIPCRVMLFMLAMNRQGSIIFLTVVAV
DRYFRVVHPHHFLNKISNRTAAIISCFLWGITIGLTVHLLYTDMMTRNGDANLCSSFSIC
YTFRWHDAMFLLEFFLPLGIILFCSGRIIWSLRQRQMDRHVKIKRAINFIMVVAIVFVIC
FLPSVAVRIRIFWLLYKHNVRNCDIYSSVDLAFFTTLSFTYMNSMLDPVVYYFSSPSFPN
FFSTCINRCLRRKTLGEPDNNRSTSVELTGDPSTIRSIPGALMTDPSEPGSPPYLASTSR
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  Blast E-value cutoff:
BDBM50211363
n/a
NameBDBM50211363
Synonyms:3-isopropyl-1H-pyrazole-5-carboxylic acid | 5-Isopropyl-1H-pyrazole-3-carboxylic acid | 5-isopropyl-3-carboxyl-pyrazole | CHEMBL238002
TypeSmall organic molecule
Emp. Form.C7H10N2O2
Mol. Mass.154.1665
SMILESCC(C)c1cc(n[nH]1)C(O)=O
Structure
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