| Reaction Details |
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 | Report a problem with these data |
| Target | Prostaglandin E2 receptor EP1 subtype |
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| Ligand | BDBM50150977 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_302495 (CHEMBL828212) |
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| Ki | 3800±n/a nM |
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| Citation |  Torisu, K; Kobayashi, K; Iwahashi, M; Egashira, H; Nakai, Y; Okada, Y; Nanbu, F; Ohuchida, S; Nakai, H; Toda, M Discovery of new chemical leads for prostaglandin D2 receptor antagonists. Bioorg Med Chem Lett14:4557-62 (2004) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Prostaglandin E2 receptor EP1 subtype |
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| Name: | Prostaglandin E2 receptor EP1 subtype |
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| Synonyms: | PE2R1_MOUSE | PGE receptor, EP1 subtype | Prostaglandin E1 | Prostaglandin E2 receptor EP1 subtype | Prostanoid EP1 receptor | Ptger1 | Ptgerep1 |
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| Type: | G-protein coupled receptor |
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| Mol. Mass.: | 43000.62 |
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| Organism: | Mus musculus (Mouse) |
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| Description: | n/a |
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| Residue: | 405 |
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| Sequence: | MSPCGLNLSLADEAATCATPRLPNTSVVLPTGDNGTSPALPIFSMTLGAVSNVLALALLA
QVAGRMRRRRSAATFLLFVASLLAIDLAGHVIPGALVLRLYTAGRAPAGGACHFLGGCMV
FFGLCPLLLGCGMAVERCVGVTQPLIHAARVSVARARLALAVLAAMALAVALLPLVHVGR
YELQYPGTWCFISLGPRGGWRQALLAGLFAGLGLAALLAALVCNTLSGLALLRARWRRRR
SRRFRKTAGPDDRRRWGSRGPRLASASSASSITSATATLRSSRGGGSARRVHAHDVEMVG
QLVGIMVVSCICWSPLLVLVVLAIGGWNSNSLQRPLFLAVRLASWNQILDPWVYILLRQA
MLRQLLRLLPLRVSAKGGPTELGLTKSAWEASSLRSSRHSGFSHL
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| BDBM50150977 |
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| n/a |
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| Name | BDBM50150977 |
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| Synonyms: | 1-(4-Butoxy-benzoyl)-5-methoxy-2-propyl-1H-indole-3-carboxylic acid | CHEMBL186244 |
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| Type | Small organic molecule |
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| Emp. Form. | C24H27NO5 |
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| Mol. Mass. | 409.4749 |
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| SMILES | CCCCOc1ccc(cc1)C(=O)n1c(CCC)c(C(O)=O)c2cc(OC)ccc12 |
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| Structure | 
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