| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Somatostatin receptor type 5 |
|---|
| Ligand | BDBM50169469 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_302433 (CHEMBL827131) |
|---|
| Ki | 7.8±n/a nM |
|---|
| Citation |  Contour-Galcéra, MO; Sidhu, A; Plas, P; Roubert, P 3-Thio-1,2,4-triazoles, novel somatostatin sst2/sst5 agonists. Bioorg Med Chem Lett15:3555-9 (2005) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Somatostatin receptor type 5 |
|---|
| Name: | Somatostatin receptor type 5 |
|---|
| Synonyms: | SOMATOSTATIN SST5 | SS-5-R | SS5-R | SS5R | SSR5_HUMAN | SSTR5 | Somatostatin receptor type 5 (SSTR5) |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 39218.02 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P35346 |
|---|
| Residue: | 364 |
|---|
| Sequence: | MEPLFPASTPSWNASSPGAASGGGDNRTLVGPAPSAGARAVLVPVLYLLVCAAGLGGNTL
VIYVVLRFAKMKTVTNIYILNLAVADVLYMLGLPFLATQNAASFWPFGPVLCRLVMTLDG
VNQFTSVFCLTVMSVDRYLAVVHPLSSARWRRPRVAKLASAAAWVLSLCMSLPLLVFADV
QEGGTCNASWPEPVGLWGAVFIIYTAVLGFFAPLLVICLCYLLIVVKVRAAGVRVGCVRR
RSERKVTRMVLVVVLVFAGCWLPFFTVNIVNLAVALPQEPASAGLYFFVVILSYANSCAN
PVLYGFLSDNFRQSFQKVLCLRKGSGAKDADATEPRPDRIRQQQEATPPAHRAAANGLMQ
TSKL
|
|
|
|---|
| BDBM50169469 |
|---|
| n/a |
|---|
| Name | BDBM50169469 |
|---|
| Synonyms: | 4-{3-(6-Fluoro-quinolin-2-yl)-5-[2-(1H-indol-3-yl)-ethylsulfanyl]-[1,2,4]triazol-4-yl}-butylamine | CHEMBL364418 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C25H25FN6S |
|---|
| Mol. Mass. | 460.57 |
|---|
| SMILES | NCCCCn1c(SCCc2c[nH]c3ccccc23)nnc1-c1ccc2cc(F)ccc2n1 |
|---|
| Structure | 
|
|---|
Search and Browse
