| Reaction Details |
|---|
 | Report a problem with these data |
| Target | P2Y purinoceptor 6 |
|---|
| Ligand | BDBM50199174 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_413300 (CHEMBL911821) |
|---|
| EC50 | >100000±n/a nM |
|---|
| Citation |  El-Tayeb, A; Qi, A; Müller, CE Synthesis and structure-activity relationships of uracil nucleotide derivatives and analogues as agonists at human P2Y2, P2Y4, and P2Y6 receptors. J Med Chem49:7076-87 (2006) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| P2Y purinoceptor 6 |
|---|
| Name: | P2Y purinoceptor 6 |
|---|
| Synonyms: | P2RY6 | P2RY6_HUMAN | P2Y purinoceptor 6 | P2Y6 | Pyrimidinergic receptor P2Y6 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 36452.29 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_1511151 |
|---|
| Residue: | 328 |
|---|
| Sequence: | MEWDNGTGQALGLPPTTCVYRENFKQLLLPPVYSAVLAAGLPLNICVITQICTSRRALTR
TAVYTLNLALADLLYACSLPLLIYNYAQGDHWPFGDFACRLVRFLFYANLHGSILFLTCI
SFQRYLGICHPLAPWHKRGGRRAAWLVCVAVWLAVTTQCLPTAIFAATGIQRNRTVCYDL
SPPALATHYMPYGMALTVIGFLLPFAALLACYCLLACRLCRQDGPAEPVAQERRGKAARM
AVVVAAAFAISFLPFHITKTAYLAVRSTPGVPCTVLEAFAAAYKGTRPFASANSVLDPIL
FYFTQKKFRRRPHELLQKLTAKWQRQGR
|
|
|
|---|
| BDBM50199174 |
|---|
| n/a |
|---|
| Name | BDBM50199174 |
|---|
| Synonyms: | 3-phenacyl-1-beta-D-ribofuranosylpyrimidine-2,4-dione 5'-monophosphate | CHEMBL215381 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C17H19N2O10P |
|---|
| Mol. Mass. | 442.3139 |
|---|
| SMILES | O[C@H]1[C@@H](O)[C@@H](O[C@@H]1COP(O)(O)=O)n1ccc(=O)n(CC(=O)c2ccccc2)c1=O |
|---|
| Structure | 
|
|---|
Search and Browse
