| Reaction Details |
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 | Report a problem with these data |
| Target | Quorum-sensing transcriptional repressor QscR |
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| Ligand | BDBM50351511 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_466841 (CHEMBL925889) |
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| EC50 | 11±n/a nM |
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| Citation |  Mattmann, ME; Geske, GD; Worzalla, GA; Chandler, JR; Sappington, KJ; Greenberg, EP; Blackwell, HE Synthetic ligands that activate and inhibit a quorum-sensing regulator in Pseudomonas aeruginosa. Bioorg Med Chem Lett18:3072-5 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Quorum-sensing transcriptional repressor QscR |
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| Name: | Quorum-sensing transcriptional repressor QscR |
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| Synonyms: | PhzR |
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| Type: | PROTEIN |
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| Mol. Mass.: | 27251.33 |
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| Organism: | Pseudomonas aeruginosa |
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| Description: | ChEMBL_466843 |
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| Residue: | 237 |
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| Sequence: | MHDEREGYLEILSRITTEEEFFSLVLEICGNYGFEFFSFGARAPFPLTAPKYHFLSNYPG
EWKSRYISEDYTSIDPIVRHGLLEYTPLIWNGEDFQENRFFWEEALHHGIRHGWSIPVRG
KYGLISMLSLVRSSESIAATEILEKESFLLWITSMLQATFGDLLAPRIVPESNVRLTARE
TEMLKWTAVGKTYGEIGLILSIDQRTVKFHIVNAMRKLNSSNKAEATMKAYAIGLLN
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| BDBM50351511 |
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| n/a |
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| Name | BDBM50351511 |
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| Synonyms: | CHEMBL463321 |
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| Type | Small organic molecule |
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| Emp. Form. | C12H19NO4 |
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| Mol. Mass. | 241.2836 |
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| SMILES | CCCCCC(=O)CC(=O)N[C@H]1CCOC1=O |r| |
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| Structure | 
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