Reaction Details | |||
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Target | Cyclin-dependent kinase 5 activator 1 | ||
Ligand | BDBM50132003 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | ChEMBL_473638 (CHEMBL937655) | ||
IC50 | 100±n/a nM | ||
Citation | Fedorov, O; Marsden, B; Pogacic, V; Rellos, P; Müller, S; Bullock, AN; Schwaller, J; Sundström, M; Knapp, S A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases. Proc Natl Acad Sci U S A104:20523-8 (2007) [PubMed] Article | ||
More Info.: | Get all data from this article, Assay Method | ||
Cyclin-dependent kinase 5 activator 1 | |||
Name: | Cyclin-dependent kinase 5 activator 1 | ||
Synonyms: | CD5R1_HUMAN | CDK5R | CDK5R1 | Cyclin-Dependent Kinase 5 Activator 1, p35 | Cyclin-dependent kinase 5 (CDK5/p25) | Cyclin-dependent kinase 5 regulatory subunit 1 | NCK5A | TPKII regulatory subunit | p35 | ||
Type: | Enzyme Subunit | ||
Mol. Mass.: | 34077.43 | ||
Organism: | Homo sapiens (Human) | ||
Description: | Q15078 | ||
Residue: | 307 | ||
Sequence: |
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BDBM50132003 | |||
n/a | |||
Name | BDBM50132003 | ||
Synonyms: | (Z)-1H,1''H-[2,3'']Biindolylidene-3,2''-dione 3-oxime | (Z)-1H,1'H-[2,3']Biindolylidene-3,2'-dione 3-oxime | 1H,1''H-[2,3'']Biindolylidene-3,2''-dione 3-oxime | 1H,1'H-[2,3']Biindolylidene-3,2'-dione 3-oxime | 3-(3-(hydroxyimino)indolin-2-ylidene)indolin-2-one | CHEMBL126077 | ||
Type | Small organic molecule | ||
Emp. Form. | C16H11N3O2 | ||
Mol. Mass. | 277.2774 | ||
SMILES | Oc1[nH]c2ccccc2c1-c1[nH]c2ccccc2c1N=O |(1.71,2.82,;2.18,1.35,;3.65,.86,;3.62,-.68,;4.77,-1.7,;4.44,-3.2,;2.97,-3.66,;1.85,-2.62,;2.18,-1.13,;1.27,.12,;-.27,.12,;-1.18,-1.12,;-2.65,-.64,;-3.96,-1.41,;-5.29,-.64,;-5.29,.9,;-3.96,1.68,;-2.63,.9,;-1.16,1.38,;-.69,2.84,;-1.7,3.98,)| | ||
Structure |