| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A2a |
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| Ligand | BDBM50207817 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_529842 (CHEMBL967545) |
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| Ki | 4920±n/a nM |
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| Citation |  Ishiyama, H; Ohshita, K; Abe, T; Nakata, H; Kobayashi, J Synthesis of eudistomin D analogues and its effects on adenosine receptors. Bioorg Med Chem16:3825-30 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A2a |
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| Name: | Adenosine receptor A2a |
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| Synonyms: | A2A adenosine receptor (hA2A) | AA2AR_HUMAN | ADENOSINE A2 | ADENOSINE A2a | ADORA2 | ADORA2A | Adenosine A2A receptor (A2AAR) |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 44716.46 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P29274 |
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| Residue: | 412 |
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| Sequence: | MPIMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADIAVGVLAI
PFAITISTGFCAACHGCLFIACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGTR
AKGIIAICWVLSFAIGLTPMLGWNNCGQPKEGKNHSQGCGEGQVACLFEDVVPMNYMVYF
NFFACVLVPLLLMLGVYLRIFLAARRQLKQMESQPLPGERARSTLQKEVHAAKSLAIIVG
LFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFR
KIIRSHVLRQQEPFKAAGTSARVLAAHGSDGEQVSLRLNGHPPGVWANGSAPHPERRPNG
YALGLVSGGSAQESQGNTGLPDVELLSHELKGVCPEPPGLDDPLAQDGAGVS
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| BDBM50207817 |
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| n/a |
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| Name | BDBM50207817 |
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| Synonyms: | 5,7-dibromo-9H-pyrido[3,4-b]indol-6-ol | 7-bromo-eudistomin D | CHEMBL272185 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H6Br2N2O |
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| Mol. Mass. | 341.986 |
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| SMILES | Oc1c(Br)cc2[nH]c3cnccc3c2c1Br |
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| Structure | 
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