| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A1 |
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| Ligand | BDBM50259665 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_527328 (CHEMBL972848) |
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| Ki | >50000±n/a nM |
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| Citation |  Ingkaninan, K; IJzerman, AP; Verpoorte, R Luteolin, a compound with adenosine A(1) receptor-binding activity, and chromone and dihydronaphthalenone constituents from Senna siamea. J Nat Prod63:315-7 (2000) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A1 |
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| Name: | Adenosine receptor A1 |
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| Synonyms: | AA1R_RAT | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | Adenosine A1 receptor (A1) | Adenosine receptor | Adenosine receptors A1 | Adora1 |
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| Type: | Protein |
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| Mol. Mass.: | 36704.13 |
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| Organism: | Rattus norvegicus (rat) |
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| Description: | n/a |
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| Residue: | 326 |
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| Sequence: | MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVT
QRRAAVAIAGCWILSLVVGLTPMFGWNNLSVVEQDWRANGSVGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALIL
FLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFL
KIWNDHFRCQPKPPIDEDLPEEKAED
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| BDBM50259665 |
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| n/a |
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| Name | BDBM50259665 |
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| Synonyms: | 5-acetonyl-7-hydroxy-2-hydroxymethylchromone | CHEMBL449531 |
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| Type | Small organic molecule |
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| Emp. Form. | C13H12O5 |
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| Mol. Mass. | 248.2314 |
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| SMILES | CC(=O)Cc1cc(O)cc2oc(CO)cc(=O)c12 |
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| Structure | 
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