Reaction Details | |||
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Target | Small conductance calcium-activated potassium channel protein 3 | ||
Ligand | BDBM50061977 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | ChEMBL_494975 (CHEMBL1008047) | ||
Kd | 2.7±n/a nM | ||
Citation | Sørensen, US; Strøbaek, D; Christophersen, P; Hougaard, C; Jensen, ML; Nielsen, EŘ; Peters, D; Teuber, L Synthesis and structure-activity relationship studies of 2-(N-substituted)-aminobenzimidazoles as potent negative gating modulators ofsmall conductance Ca2+-activated K+ channels. J Med Chem51:7625-34 (2009) [PubMed] Article | ||
More Info.: | Get all data from this article, Assay Method | ||
Small conductance calcium-activated potassium channel protein 3 | |||
Name: | Small conductance calcium-activated potassium channel protein 3 | ||
Synonyms: | KCNN3_RAT | Kcnn3 | SK3 | Small conductance calcium-activated potassium channel | ||
Type: | PROTEIN | ||
Mol. Mass.: | 81476.29 | ||
Organism: | Rattus norvegicus | ||
Description: | ChEMBL_494975 | ||
Residue: | 732 | ||
Sequence: |
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BDBM50061977 | |||
n/a | |||
Name | BDBM50061977 | ||
Synonyms: | 17,25-diazonia-2,9-diazaheptacyclo[23.6.2.24,7.210,17.119,23.011,16.026,31]octatriaconta-1(31),4,6,10(35),11,13,15,17(34),19,21,23(38),25,27,29,32,36-hexadecaene | 17,25-diazonia-2,9-diazaheptacyclo[23.6.2.24,7.210,17.119,23.011,16.026,31]octatriaconta-1(32),4,6,10(35),11(16),12,14,17(34),19,21,23(38),25(33),26(31),27,29,36-hexadecaene | CHEMBL117908 | CHEMBL45193 | UCL-1684 | ||
Type | Small organic molecule | ||
Emp. Form. | C34H30N4 | ||
Mol. Mass. | 494.6277 | ||
SMILES | C1N[c+]2ccn(Cc3cccc(Cn4cc[c+](NCc5ccc1cc5)c1ccccc41)c3)c1ccccc21 | ||
Structure |