| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM50296142 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_579534 (CHEMBL1059681) |
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| Ki | 3919±n/a nM |
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| Citation |  Foloppe, N; Benwell, K; Brooks, TD; Kennett, G; Knight, AR; Misra, A; Monck, NJ Discovery and functional evaluation of diverse novel human CB(1) receptor ligands. Bioorg Med Chem Lett19:4183-90 (2009) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 39690.94 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P34972 |
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| Residue: | 360 |
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| Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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| BDBM50296142 |
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| n/a |
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| Name | BDBM50296142 |
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| Synonyms: | 1-(1-(4-chlorophenyl)-4-(3-methoxyphenyl)-5-(4-morpholinophenyl)-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethanone | CHEMBL554943 |
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| Type | Small organic molecule |
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| Emp. Form. | C27H27ClN4O3 |
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| Mol. Mass. | 490.981 |
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| SMILES | COc1cccc(c1)N1C(N(N=C1C(C)=O)c1ccc(Cl)cc1)c1ccc(cc1)N1CCOCC1 |c:12| |
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| Structure | 
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