| Reaction Details |
|---|
 | Report a problem with these data |
| Target | P2Y purinoceptor 2 |
|---|
| Ligand | BDBM50378128 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_587770 (CHEMBL1040421) |
|---|
| IC50 | 264000±n/a nM |
|---|
| Citation |  Sauer, R; El-Tayeb, A; Kaulich, M; Müller, CE Synthesis of uracil nucleotide analogs with a modified, acyclic ribose moiety as P2Y(2) receptor antagonists. Bioorg Med Chem17:5071-9 (2009) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| P2Y purinoceptor 2 |
|---|
| Name: | P2Y purinoceptor 2 |
|---|
| Synonyms: | ATP receptor | P2RY2_MOUSE | P2U purinoceptor 1 | P2U1 | P2Y purinoceptor 2 | P2Y2 | P2ru1 | P2ry2 | Purinergic receptor | Purinergic receptor P2Y2 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 42202.78 |
|---|
| Organism: | Mus musculus |
|---|
| Description: | ChEMBL_587770 |
|---|
| Residue: | 373 |
|---|
| Sequence: | MAADLEPWNSTINGTWEGDELGYKCRFNEDFKYVLLPVSYGVVCVLGLCLNVVALYIFLC
RLKTWNASTTYMFHLAVSDSLYAASLPLLVYYYARGDHWPFSTVLCKLVRFLFYTNLYCS
ILFLTCISVHRCLGVLRPLHSLRWGRARYARRVAAVVWVLVLACQAPVLYFVTTSVRGTR
ITCHDTSARELFSHFVAYSSVMLGLLFAVPFSVILVCYVLMARRLLKPAYGTTGGLPRAK
RKSVRTIALVLAVFALCFLPFHVTRTLYYSFRSLDLSCHTLNAINMAYKITRPLASANSC
LDPVLYFLAGQRLVRFARDAKPPTEPTPSPQARRKLGLHRPNRTVRKDLSVSSDDSRRTE
STPAGSETKDIRL
|
|
|
|---|
| BDBM50378128 |
|---|
| n/a |
|---|
| Name | BDBM50378128 |
|---|
| Synonyms: | CHEMBL575653 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C8H15N2O13P3 |
|---|
| Mol. Mass. | 440.1316 |
|---|
| SMILES | OP(O)(=O)OP(O)(=O)OP(O)(=O)OCCCOCn1ccc(=O)[nH]c1=O |
|---|
| Structure | 
|
|---|
Search and Browse
