| Reaction Details |
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 | Report a problem with these data |
| Target | P2Y purinoceptor 4 |
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| Ligand | BDBM50268876 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_718669 (CHEMBL1680820) |
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| IC50 | >10000±n/a nM |
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| Citation |  Baqi, Y; Hausmann, R; Rosefort, C; Rettinger, J; Schmalzing, G; Müller, CE Discovery of potent competitive antagonists and positive modulators of the P2X2 receptor. J Med Chem54:817-30 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| P2Y purinoceptor 4 |
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| Name: | P2Y purinoceptor 4 |
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| Synonyms: | NRU | P2P | P2RY4 | P2RY4_HUMAN | P2Y purinoceptor 4 | P2Y4 | Pyrimidinergic receptor P2Y4 | UNR | Uridine nucleotide receptor |
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| Type: | PROTEIN |
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| Mol. Mass.: | 40977.17 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_751027 |
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| Residue: | 365 |
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| Sequence: | MASTESSLLRSLGLSPGPGSSEVELDCWFDEDFKFILLPVSYAVVFVLGLGLNAPTLWLF
IFRLRPWDATATYMFHLALSDTLYVLSLPTLIYYYAAHNHWPFGTEICKFVRFLFYWNLY
CSVLFLTCISVHRYLGICHPLRALRWGRPRLAGLLCLAVWLVVAGCLVPNLFFVTTSNKG
TTVLCHDTTRPEEFDHYVHFSSAVMGLLFGVPCLVTLVCYGLMARRLYQPLPGSAQSSSR
LRSLRTIAVVLTVFAVCFVPFHITRTIYYLARLLEADCRVLNIVNVVYKVTRPLASANSC
LDPVLYLLTGDKYRRQLRQLCGGGKPQPRTAASSLALVSLPEDSSCRWAATPQDSSCSTP
RADRL
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| BDBM50268876 |
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| n/a |
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| Name | BDBM50268876 |
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| Synonyms: | CHEMBL509572 | Disodium 1-amino-4-[4-(4-chloro-6-methoxy-[1,3,5]triazine-2-ylamino)-3-sulfophenylamino]-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate |
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| Type | Small organic molecule |
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| Emp. Form. | C24H15ClN6O9S2 |
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| Mol. Mass. | 630.995 |
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| SMILES | COc1nc(Cl)nc(Nc2ccc(Nc3cc(c(N)c4C(=O)c5ccccc5C(=O)c34)S([O-])(=O)=O)cc2S([O-])(=O)=O)n1 |
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| Structure | 
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