| Reaction Details |
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 | Report a problem with these data |
| Target | Vesicular acetylcholine transporter |
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| Ligand | BDBM50389432 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_832035 (CHEMBL2065331) |
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| Kd | 1.73±n/a nM |
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| Citation |  Kozaka, T; Uno, I; Kitamura, Y; Miwa, D; Ogawa, K; Shiba, K Syntheses and in vitro evaluation of decalinvesamicol analogues as potential imaging probes for vesicular acetylcholine transporter (VAChT). Bioorg Med Chem20:4936-41 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Vesicular acetylcholine transporter |
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| Name: | Vesicular acetylcholine transporter |
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| Synonyms: | Slc18a3 | Solute carrier family 18 member 3 | VACHT_RAT | Vacht | Vat | rVAT |
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| Type: | PROTEIN |
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| Mol. Mass.: | 56533.41 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_1503353 |
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| Residue: | 530 |
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| Sequence: | MEPTAPTGQARAAATKLSEAVGAALQEPQRQRRLVLVIVCVALLLDNMLYMVIVPIVPDY
IAHMRGGSEGPTLVSEVWEPTLPPPTLANASAYLANTSASPTAAGSARSILRPRYPTESE
DVKIGVLFASKAILQLLVNPLSGPFIDRMSYDVPLLIGLGVMFASTVMFAFAEDYATLFA
ARSLQGLGSAFADTSGIAMIADKYPEEPERSRALGVALAFISFGSLVAPPFGGILYEFAG
KRVPFLVLAAVSLFDALLLLAVAKPFSAAARARANLPVGTPIHRLMLDPYIAVVAGALTT
CNIPLAFLEPTIATWMKHTMAASEWEMGMVWLPAFVPHVLGVYLTVRLAARYPHLQWLYG
ALGLAVIGVSSCVVPACRSFAPLVVSLCGLCFGIALVDTALLPTLAFLVDVRHVSVYGSV
YAIADISYSVAYALGPIVAGHIVHSLGFEQLSLGMGLANLLYAPVLLLLRNVGLLTRSRS
ERDVLLDEPPQGLYDAVRLREVQGKDGGEPCSPPGPFDGCEDDYNYYSRS
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| BDBM50389432 |
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| n/a |
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| Name | BDBM50389432 |
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| Synonyms: | CHEMBL2064618 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H30INO |
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| Mol. Mass. | 439.3735 |
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| SMILES | OC1C[C@@H]2CCCC[C@H]2CC1N1CCC(CC1)c1ccccc1I |r| |
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| Structure | 
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