| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Solute carrier organic anion transporter family member 2B1 |
|---|
| Ligand | BDBM50391000 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_836587 (CHEMBL2077328) |
|---|
| Ki | 3000±n/a nM |
|---|
| Citation |  Vavricka, SR; Van Montfoort, J; Ha, HR; Meier, PJ; Fattinger, K Interactions of rifamycin SV and rifampicin with organic anion uptake systems of human liver. Hepatology36:164-72 (2002) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Solute carrier organic anion transporter family member 2B1 |
|---|
| Name: | Solute carrier organic anion transporter family member 2B1 |
|---|
| Synonyms: | KIAA0880 | OATP-B | OATP-RP2 | OATP2B1 | OATPB | OATPRP2 | Organic anion transporter B | Organic anion transporter polypeptide-related protein 2 | SLC21A9 | SLCO2B1 | SO2B1_HUMAN | Solute carrier family 21 member 9 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 76729.07 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_1488531 |
|---|
| Residue: | 709 |
|---|
| Sequence: | MGPRIGPAGEVPQVPDKETKATMGTENTPGGKASPDPQDVRPSVFHNIKLFVLCHSLLQL
AQLMISGYLKSSISTVEKRFGLSSQTSGLLASFNEVGNTALIVFVSYFGSRVHRPRMIGY
GAILVALAGLLMTLPHFISEPYRYDNTSPEDMPQDFKASLCLPTTSAPASAPSNGNCSSY
TETQHLSVVGIMFVAQTLLGVGGVPIQPFGISYIDDFAHNSNSPLYLGILFAVTMMGPGL
AFGLGSLMLRLYVDINQMPEGGISLTIKDPRWVGAWWLGFLIAAGAVALAAIPYFFFPKE
MPKEKRELQFRRKVLAVTDSPARKGKDSPSKQSPGESTKKQDGLVQIAPNLTVIQFIKVF
PRVLLQTLRHPIFLLVVLSQVCLSSMAAGMAIFLPKFLERQFSITASYANLLIGCLSFPS
VIVGIVVGGVLVKRLHLGPVGCGALCLLGMLLCLFFSLPLFFIGCSSHQIAGITHQTSAH
PGLELSPSCMEACSCPLDGFNPVCDPSTRVEYITPCHAGCSSWVVQDALDNSQVFYTNCS
CVVEGNPVLAGSCDSTCSHLVVPFLLLVSLGSALACLTHTPSFMLILRGVKKEDKTLAVG
IQFMFLRILAWMPSPVIHGSAIDTTCVHWALSCGRRAVCRYYNNDLLRNRFIGLQFFFKT
GSVICFALVLAVLRQQDKEARTKESRSSPAVEQQLLVSGPGKKPEDSRV
|
|
|
|---|
| BDBM50391000 |
|---|
| n/a |
|---|
| Name | BDBM50391000 |
|---|
| Synonyms: | CB-01-11 | RIFAMYCIN |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C37H47NO12 |
|---|
| Mol. Mass. | 697.7686 |
|---|
| SMILES | CO[C@H]1\C=C\O[C@@]2(C)Oc3c(C2=O)c2c(O)cc(NC(=O)\C(C)=C/C=C/[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C)c(O)c2c(O)c3C |r,c:23,t:3,25| |
|---|
| Structure | 
|
|---|
Search and Browse
