| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
|---|
| Ligand | BDBM50399281 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_877094 (CHEMBL2186830) |
|---|
| Ki | 698±n/a nM |
|---|
| Citation |  Alapafuja, SO; Nikas, SP; Bharathan, IT; Shukla, VG; Nasr, ML; Bowman, AL; Zvonok, N; Li, J; Shi, X; Engen, JR; Makriyannis, A Sulfonyl fluoride inhibitors of fatty acid amide hydrolase. J Med Chem55:10074-89 (2012) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Cannabinoid receptor 2 |
|---|
| Name: | Cannabinoid receptor 2 |
|---|
| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CNR2_MOUSE | Cannabinoid CB2 receptor | Cannabinoid receptor | Cannabinoid receptor 2 | Cnr2 | mCB2 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 38220.43 |
|---|
| Organism: | MOUSE |
|---|
| Description: | P47936 |
|---|
| Residue: | 347 |
|---|
| Sequence: | MEGCRETEVTNGSNGGLEFNPMKEYMILSSGQQIAVAVLCTLMGLLSALENMAVLYIILS
SRRLRRKPSYLFISSLAGADFLASVIFACNFVIFHVFHGVDSNAIFLLKIGSVTMTFTAS
VGSLLLTAVDRYLCLCYPPTYKALVTRGRALVALCVMWVLSALISYLPLMGWTCCPSPCS
ELFPLIPNDYLLGWLLFIAILFSGIIYTYGYVLWKAHRHVATLAEHQDRQVPGIARMRLD
VRLAKTLGLVLAVLLICWFPALALMGHSLVTTLSDQVKEAFAFCSMLCLVNSMVNPIIYA
LRSGEIRSAAQHCLIGWKKYLQGLGPEGKEEGPRSSVTETEADVKTT
|
|
|
|---|
| BDBM50399281 |
|---|
| n/a |
|---|
| Name | BDBM50399281 |
|---|
| Synonyms: | CHEMBL2180818 | US9102622, 14.1 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C13H19FO3S |
|---|
| Mol. Mass. | 274.352 |
|---|
| SMILES | Oc1ccc(CCCCCCCS(F)(=O)=O)cc1 |
|---|
| Structure | 
|
|---|
Search and Browse
